| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| C5AR1 |
H-His-Lys-AspMet-GIn-Leu-Gly-Arg-OH |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| C5AR1 |
Tyr-Ser-Phe-Lys-Asp-cyclo[Cys-Pro-Leu-Cys]-Arg |
NA |
NA |
NA |
500000 |
NA |
NA |
TTD |
| C5AR1 |
H-His(1Me)-Lys-AspMet-GIn-Leu-Gly-Arg-OH |
180000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| C5AR1 |
2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionylamino]-6-amino-hexanoylamino}-3-carboxy-propionylamino)-4-methylsulfanyl-butyrylamino]-4-carbamoyl-butyrylamino}-4-methyl-pentanoylamino)-acetylamino]-5-guanidino-pentanoic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
Pyrophosphoric acid |
25800000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CA1 |
(1R,2R,5S,6S)-2,5-dicyclohexyl-3,4,7-trioxabicyclo[4.1.0]heptane |
950000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
Sulfamic acid isopropyl ester |
690000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
6,7-Dihydroxy-3-phenylchromen-2-one |
NA |
124000|160000 |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
Sodium Carbonate |
15000000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CA1 |
Tyrosol |
430000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| CA1 |
Propionate ion |
1010000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
Hydrogen sulfite |
18000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
Chlorate ion |
540000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
Butanoate |
511000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
4-[2-(2,4-Diphenyl-6-propylpyridin-1-ium-1-yl)ethyl]benzenesulfonamide;perchlorate |
112000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
2,4-Diphenyl-6-propyl-1-[2-(4-sulfamoyl-phenyl)-ethyl]-pyridinium; perchlorate |
112000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
4-{2-[(Trifluoromethyl)sulfonyl]hydrazino}benzenesulfonamide |
155500 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
4-[2-(2-Butyl-4,6-diphenylpyridin-1-ium-1-yl)ethyl]benzenesulfonamide;perchlorate |
290000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
2-Butyl-4,6-diphenyl-1-[2-(4-sulfamoyl-phenyl)-ethyl]-pyridinium; perchlorate |
290000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
6-Methoxy-9-phenyl-1,10-diazatricyclo[6.4.1.04,13]trideca-4(13),5,7,9-tetraen-12-one |
107000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |