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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CA1 2-[(4-fluorobenzoyl)amino]-N-(4-methyl-2-oxochromen-7-yl)benzamide 500000 NA NA NA NA NA TTD
CA1 2-[(4-chlorobenzoyl)amino]-N-[2-oxo-4-(trifluoromethyl)chromen-7-yl]benzamide 500000 NA NA NA NA NA TTD
CA1 4-Hydroxybenzoic acid 1061000 NA NA NA NA NA BindingDB
CA1 4-Hydroxyquinazoline 500000 NA NA NA NA NA TTD
CA1 2-amino-4-(3,4-dihydroxybenzylidene)-1H-imidazol-5(4H)-one 355000 NA NA NA NA NA TTD
CA1 N-(benzimidazol-1-yl)-2,4-dichloro-5-sulfamoyl-benzamide NA NA 200000 NA NA NA BindingDB
CA1 Perrhenate 110000 NA NA NA NA NA BindingDB|TTD
CA1 Sodium hexafluoroarsenate 300000000 NA NA NA NA NA TTD
CA1 Metasilicic acid 570000 NA NA NA NA NA TTD
CA1 2-phenyl-N-(2-phenylethylsulfamoyl)ethanamine 200000 NA NA NA NA NA TTD
CA1 N,N'-dibenzylsulfamide 200000 NA NA NA NA NA TTD
CA1 Hydrofluoric Acid 300000000 NA NA NA NA NA PubChem|TTD
CA1 methyl (2S)-2-[(2-methylpropan-2-yl)oxycarbonylsulfamoylamino]propanoate 200000 NA NA NA NA NA TTD
CA1 2-(3-Chloro-4-hydroxyphenyl)acetamide 237000 NA NA NA NA NA BindingDB|TTD
CA1 N-(1-naphthyl)ethylenediamine 500000 NA NA NA NA NA TTD
CA1 Cyclopentyl sulfamate 1000000 NA NA NA NA NA TTD
CA1 Pyrogallol tris-(methanesulfonate) 478300 NA NA NA NA NA BindingDB
CA1 6,7-Dihydroxy-3-(4-methylphenyl)-2h-chromen-2-one NA 256000|272000 NA NA NA NA BindingDB
CA1 [4-[[4-[4-[3-(Trifluoromethyl)phenyl]pyrimidin-2-yl]piperazine-1-carbonyl]amino]phenyl] sulfamate 3472900 NA NA NA NA NA BindingDB
CA1 [4-[[4-[4-(3-Methylphenyl)pyrimidin-2-yl]piperazine-1-carbonyl]amino]phenyl] sulfamate 4069900 NA NA NA NA NA BindingDB