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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CA1 [4-[[4-(2-Methylphenyl)piperazine-1-carbonyl]amino]phenyl] sulfamate 692000 NA NA NA NA NA BindingDB
CA1 [4-[[4-(1-Benzofuran-2-ylmethyl)piperazine-1-carbonyl]amino]phenyl] sulfamate 760300 NA NA NA NA NA BindingDB
CA1 [4-[(4-Decylpiperazine-1-carbonyl)amino]phenyl] sulfamate 680100 NA NA NA NA NA BindingDB
CA1 [4-[[4-[4-(3,4,5-Trimethoxyphenyl)pyrimidin-2-yl]piperazine-1-carbonyl]amino]phenyl] sulfamate 5284000 NA NA NA NA NA BindingDB
CA1 [4-[[4-[4-(4-Methoxyphenyl)pyrimidin-2-yl]piperazine-1-carbonyl]amino]phenyl] sulfamate 3930400 NA NA NA NA NA BindingDB
CA1 hCAIX-IN-3 7769100 NA NA NA NA NA BindingDB
CA1 [4-[[4-(4-Phenylpyrimidin-2-yl)piperazine-1-carbonyl]amino]phenyl] sulfamate 2370900 NA NA NA NA NA BindingDB
CA1 [4-[(4-Octylpiperazine-1-carbonyl)amino]phenyl] sulfamate 752300 NA NA NA NA NA BindingDB
CA1 [4-[[4-(3,4-Dichlorophenyl)piperazine-1-carbonyl]amino]phenyl] sulfamate 918800 NA NA NA NA NA BindingDB
CA1 N1,N2-(2-(2,2,2-Trifluoroacetamido)ethyl)ethane-1,2-diaminium Trifluoroacetate 500000 NA NA NA NA NA TTD
CA1 Carbonotrithioate 790000 NA NA NA NA NA BindingDB
CA1 Sulfosulfamic acid 310000 NA NA NA NA NA TTD
CA1 2-(3-chloro-4-hydroxyphenyl)-N-(2-methoxyethyl)acetamide 158000 NA NA NA NA NA BindingDB|TTD
CA1 4-Sulfosalicylic acid NA|480000 290000|NA NA NA NA NA BindingDB|TTD
CA1 Isobutyrate 120000 NA NA NA NA NA BindingDB
CA1 Hexafluoroaluminate(3-) 52400000 NA NA NA NA NA BindingDB
CA1 Cryolite 52400000 NA NA NA NA NA TTD
CA1 2-(benzyloxyamino)-N-hydroxy-3-methylpentanamide 435000 NA NA NA NA NA BindingDB|TTD
CA1 Periodate 14600000 NA NA NA NA NA BindingDB
CA1 Endiandrin A 368000 NA NA NA NA NA BindingDB|TTD