| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CA1 |
(1R,2S,5R,6S)-2-cyclohexyl-5-phenyl-3,4,7-trioxabicyclo[4.1.0]heptane |
124000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
|
25800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
|
540000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
|
660000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
|
640000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
|
118000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
7-(3-aminopyrrolidin-1-yl)-6-fluoro-3-[(3-phenylpropylamino)methyl]-1H-1,8-naphthyridin-4-one |
8400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
6-fluoro-3-(hydroxymethyl)-7-pyrrolidin-1-yl-1H-1,8-naphthyridin-4-one |
12000000|15000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
3-[(benzylamino)methyl]-6-fluoro-7-pyrrolidin-1-yl-1H-1,8-naphthyridin-4-one |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
6-fluoro-7-pyrrolidin-1-yl-1H-1,8-naphthyridin-4-one |
18000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
Sulfamic acid (3S,10R,17R)-17-((R)-1,5-dimethyl-hexyl)-10-methyl-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
(1R,2S,6R,8S)-4,4,11,11-tetramethyl-6-[(sulfamoylamino)carbamoyl]-3,5,7,10,12-pentaoxatricyclo[6.4.0.02,6]dodecane |
420000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
[(1R,2S,6S,8S,9R)-4,4,11,11-tetramethyl-3,5,7,10,12-pentaoxatricyclo[7.3.0.02,6]dodecan-8-yl]methyl sulfamate |
400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
CID 44391604 |
310000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
Phenoxyarsonous acid |
31700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
5-[4-(4-Bromo-benzenesulfonyl)-phenyl]-4-m-tolyl-4H-[1,2,4]triazole-3-thiol |
254000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
N-(5-Mercapto-[1,3,4]thiadiazol-2-yl)-2-nitro-benzenesulfonamide |
303000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
2,3,4,5,6-Pentafluoro-N-(5-mercapto-[1,3,4]thiadiazol-2-yl)-benzamide |
308000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
5-[4-(4-Bromo-benzenesulfonyl)-phenyl]-4-p-tolyl-4H-[1,2,4]triazole-3-thiol |
249000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
2-(aminosulfonyl)-5-chloro-4-methylphenyl-N-(4-nitrophenyl)propanehydrazonothioate |
220000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |