| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CA1 |
2-(aminosulfonyl)-5-chloro-4-methylphenyl N-(phenylsulfonyl)benzenecarbohydrazonothioate |
113000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
6-(isobutylthio)-3,4-dihydro-2H-1,2,4-benzothiadiazine-7-sulfonamide 1,1-dioxide |
392000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
6-[(1,1-dioxo-7-sulfamoyl-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-6-yl)disulfanyl]-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazine-7-sulfonamide |
310000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
2-{4-chlorobenzyloxy[(4-methoxyphenyl)sulfonyl]amino}-N-hydroxyacetamide |
156000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
2-(benzyloxyamino)-N-hydroxyacetamide |
490000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
2-(benzyloxyamino)-N-hydroxyhexanamide |
520000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
N-(Cyclopropylsulfamoyl)Cyclopropanamine |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
N,N,N',N'-tetrabutylsulfamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
1-[(E)-(2-nitrophenyl)methylideneamino]-3-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)urea |
222820 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
1-[(E)-[2-(dimethylamino)phenyl]methylideneamino]-3-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)urea |
125000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
1-[(E)-1-(4-chlorophenyl)ethylideneamino]-3-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)urea |
144070 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
(2R(S),7R(S))-7-Hydroxybicyclo[2.2.1]heptan-2-yl nitrate |
13600000|NA |
NA|7130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
Foscarnet Sodium |
24100000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CA1 |
Ferulic acid |
408000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
N-(N-Boc-sulfamoyl)glycine Methyl Ester |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
Sodium phenylarsonate |
31700000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
Sodium (Trihydroxy)phenylborate |
31700000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA1 |
Cgs-27023 |
281000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA1 |
Oxo(Phenyl)-Boranediol |
31700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA1 |
trans-(1S(R),8S(R),Z)-8-Hydroxycyclooct-4-enyl nitrate |
41800000|NA |
NA|21000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |