| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CA2 |
1-(2,4-Dichlorophenyl)-3-(4-(1,3,7,7-tetramethyl-5-oxo-1,2,3,4,5,6,7,8-octahydroquinazolin-4-yl)phenyl)thiourea (4h) |
NA |
151090 |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
N-(5-metoksi-1,2,3,4-tetrahydronaphthalene-1-yl)methanesulfonamide (30) |
112000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
2-benzamido-N-[2-oxo-4-(trifluoromethyl)chromen-7-yl]benzamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
ethyl 6-fluoro-4-oxo-7-pyrrolidin-1-yl-1H-1,8-naphthyridine-3-carboxylate |
760000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
2-[(3,4,5-trimethoxyphenyl)methyl]-3,4-dihydro-1H-isoquinolin-6-ol |
678960 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA2 |
2-[(4-fluorobenzoyl)amino]-N-[2-oxo-4-(trifluoromethyl)chromen-7-yl]benzamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
2-benzamido-N-(4-methyl-2-oxochromen-7-yl)benzamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
2-[(4-chlorobenzoyl)amino]-N-(4-methyl-2-oxochromen-7-yl)benzamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
2-[(4-fluorobenzoyl)amino]-N-(4-methyl-2-oxochromen-7-yl)benzamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
2-[(4-chlorobenzoyl)amino]-N-[2-oxo-4-(trifluoromethyl)chromen-7-yl]benzamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
4-Hydroxybenzoic acid |
675000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
4-Hydroxyquinazoline |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
1-[(E)-(4-hydroxy-3-methoxyphenyl)methylideneamino]-3-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)urea |
386000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
1-[(E)-1-(4-hydroxyphenyl)ethylideneamino]-3-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)urea |
350000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
(5Z)-5-[(2,4-dimethoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
NA |
NA |
1000000|1e+06 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| CA2 |
Perrhenate |
750000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA2 |
Sodium hexafluoroarsenate |
9400000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
Metasilicic acid |
2680000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
2-phenyl-N-(2-phenylethylsulfamoyl)ethanamine |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
Hydrofluoric Acid |
300000000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |