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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CA2 methyl (2S)-2-[(2-methylpropan-2-yl)oxycarbonylsulfamoylamino]propanoate 200000 NA NA NA NA NA TTD
CA2 4-Amino-3-chlorobenzenesulfonamide 110000|9090000 NA NA NA NA NA BindingDB
CA2 2-(3-Chloro-4-hydroxyphenyl)acetamide 131000 NA NA NA NA NA BindingDB|TTD
CA2 N-(1-naphthyl)ethylenediamine 103000 NA NA NA NA NA BindingDB|TTD
CA2 6,7-Dihydroxy-3-(4-methylphenyl)-2h-chromen-2-one NA 127000|561000 NA NA NA NA BindingDB
CA2 [4-[[4-[4-[3-(Trifluoromethyl)phenyl]pyrimidin-2-yl]piperazine-1-carbonyl]amino]phenyl] sulfamate 457700 NA NA NA NA NA BindingDB
CA2 [4-[[4-[4-(3-Methylphenyl)pyrimidin-2-yl]piperazine-1-carbonyl]amino]phenyl] sulfamate 206900|1317300 NA NA NA NA NA BindingDB
CA2 [4-[[4-(2-Methylphenyl)piperazine-1-carbonyl]amino]phenyl] sulfamate 759300 NA NA NA NA NA BindingDB
CA2 [4-[[4-(1-Benzofuran-2-ylmethyl)piperazine-1-carbonyl]amino]phenyl] sulfamate 4223000 NA NA NA NA NA BindingDB
CA2 [4-[(4-Decylpiperazine-1-carbonyl)amino]phenyl] sulfamate 4189500 NA NA NA NA NA BindingDB
CA2 [4-[[4-[4-(3,4,5-Trimethoxyphenyl)pyrimidin-2-yl]piperazine-1-carbonyl]amino]phenyl] sulfamate 279800 NA NA NA NA NA BindingDB
CA2 [4-[[4-[4-(4-Methoxyphenyl)pyrimidin-2-yl]piperazine-1-carbonyl]amino]phenyl] sulfamate 384100 NA NA NA NA NA BindingDB
CA2 hCAIX-IN-3 124200|831300 NA NA NA NA NA BindingDB
CA2 [4-[[4-(4-Phenylpyrimidin-2-yl)piperazine-1-carbonyl]amino]phenyl] sulfamate 705500|4097600 NA NA NA NA NA BindingDB
CA2 [4-[(4-Octylpiperazine-1-carbonyl)amino]phenyl] sulfamate 4797500 NA NA NA NA NA BindingDB
CA2 [4-[[4-(3,4-Dichlorophenyl)piperazine-1-carbonyl]amino]phenyl] sulfamate 1641600 NA NA NA NA NA BindingDB
CA2 Pyrithione 510000 NA NA NA NA NA BindingDB|PubChem|TTD
CA2 N,N'-dipropylsulfamide 124000 NA NA NA NA NA BindingDB|TTD
CA2 N1,N2-(2-(2,2,2-Trifluoroacetamido)ethyl)ethane-1,2-diaminium Trifluoroacetate 500000 NA NA NA NA NA TTD
CA2 Carbonotrithioate 460000 NA NA NA NA NA BindingDB