Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CA3 | 3-(2-bromophenyl)-2-(hydrazinecarbonyl)-1H-indole-5-sulfonamide | 3900000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | 3-(3-bromophenyl)-2-(hydrazinecarbonyl)-1H-indole-5-sulfonamide | 5500000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | 3-(4-bromophenyl)-2-(hydrazinecarbonyl)-1H-indole-5-sulfonamide | 5200000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | 2-(hydrazinecarbonyl)-3-(3-methoxyphenyl)-1H-indole-5-sulfonamide | 5500000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | 2-(hydrazinecarbonyl)-3-(2,3,4,5,6-pentafluorophenyl)-1H-indole-5-sulfonamide | 5400000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | Celecoxib | 154000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | 2,2,2-Trifluoro-N-(2-(naphthalen-1-ylamino)-acetamide | 128000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | Dichlorphenamide | 630000|680000|684000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | 4-((2-Amino-4-pyrimidinyl)amino)benzenesulfonamide | 2633000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | Coumarin | 200000 | NA | NA | NA | NA | NA | PubChem |
| CA3 | Ethoxzolamide | 1000000|1100000|1113000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | Salicylic Acid | 885000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | Furosemide [USAN:USP:INN:BAN:JAN] | 3200000 | NA | NA | NA | NA | NA | PubChem |
| CA3 | Indapamide | 230000 | NA | NA | NA | NA | NA | PubChem |
| CA3 | N1,N12-Bis(trifluoroacetyl)-N4,N8-bis(t-butoxycarbonyl)spermine | 112000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | Spermine(hbbh) | 132000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | N-(5-sulfamoyl-1,3,4-thiadiazol-2-yl)adamantane-1-carboxamide | 300000|310000|1200000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | Mafenide | 681000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | Methazolamide | 700000|770000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | 4-[[(4-Aminophenyl)sulfonylamino]methyl]benzenesulfonamide | 114000 | NA | NA | NA | NA | NA | BindingDB |