Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CA3 | N-(2-Fluoro-4-Sulfamoylphenyl)-2-(Thiophen-2-Yl)acetamide | 1200000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | 4-Amino-3-fluorobenzene-1-sulfonamide | 2075000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | 2-(1-adamantyl)-N-(5-sulfamoyl-1,3,4-thiadiazol-2-yl)acetamide | 410000|1400000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | Resorcinol | 605000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | 5-(1h-Benzimidazol-1-Ylacetyl)-2-Chlorobenzenesulfonamide | NA | NA | 200000 | NA | NA | NA | BindingDB |
| CA3 | Saccharin | 1000000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | 5-Imino-4-methyl-1,3,4-thiadiazole-2-sulfonamide | 198000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | Dorzolamide | 770000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | Topiramate | 780000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | Irosustat | 700000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | 1-N-(4-Sulfamoylphenyl-ethyl)-2,4,6-trimethylpyridinium | 300000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | 2-Chloro-5-[(2-methyl-1H-benzimidazol-1-yl)acetyl]benzenesulfonamide | NA | NA | 200000 | NA | NA | NA | BindingDB |
| CA3 | 2-Chloro-5-[(2-ethyl-1H-benzimidazol-1-yl)acetyl]benzenesulfonamide | NA | NA | 125000 | NA | NA | NA | BindingDB |
| CA3 | Sulfanilamide | 988000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | Sulthiame | 630000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | Investigational agent, 5 | 330000 | NA | NA | NA | NA | NA | BindingDB |
| CA3 | Trichlormethiazide | 560000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | Zonisamide | 2200000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| CA3 | 2,4-dichloro-N-cyclohexyl-5-sulfamoylbenzamide | NA | NA | 200000 | NA | NA | NA | BindingDB |
| CA3 | N-(4-sulfamoylphenyl)-2-(thiophen-2-yl)acetamide | 800000 | NA | NA | NA | NA | NA | BindingDB |