| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CAMK2G |
R-K-K-Y-K-K-R-R-K-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CAMK2G |
R-K-K-Y-K-G-R-R-K-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CAMK2G |
R-K-K-(Ach)-(Ach)-(Ach)-R-R-K-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CAMK2G |
R-K-K-(Ach)-K-(Ach)-R-R-K-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CAMK2G |
R-K-K-(Ach)-K-Y-R-R-K-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CAMK2G |
R-K-K-(Ach)-(Ach)-Y-R-R-K-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CAMK2G |
R-K-K-Y-(Ach)-(Ach)-R-R-K-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CAMK2G |
R-K-K-Y-K-(Ach)-R-R-K-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CAMK2G |
H-Arg-Lys-Lys-Tyr-Lys-aThr-Arg-Arg-Lys-NH2 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CAMK2G |
10-Chloro-6-hydroxy-11lambda5-pyrido(1,2-A)quinolin-11-ylium chloride |
NA |
760000 |
NA |
NA |
NA |
NA |
TTD |
| CANX |
2-[2-[[(1S,2S,3S,4R,5S)-2,4-dihydroxy-5-(hydroxymethyl)-3-[(2R,3S,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxycyclohexyl]oxycarbonylamino]ethoxy]ethyl N-[[1,3-bis[2-[[(2R,3R,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxycarbonylamino]ethoxycarbonylamino]propan-2-yloxycarbonylamino]-hydroxymethyl]carbamate |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
| CAPN1 |
N-(4-fluorophenylsulfonyl)-D-valyl-D-leucinal |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CAPN1 |
[2-[(E)-[2-methylpropyl-[2-[2-methylpropyl(phenylmethoxycarbonylamino)amino]-2-oxoethyl]hydrazinylidene]methyl]phenyl]boronic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CAPN1 |
[3-[(E)-[benzyl-[2-[2-methylpropyl(phenylmethoxycarbonylamino)amino]-2-oxoethyl]hydrazinylidene]methyl]phenyl]boronic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CAPN1 |
N-[4-(ethylamino)-3,4-dioxo-1-phenylbutan-2-yl]-1-naphthalen-2-ylsulfonylpiperidine-4-carboxamide |
800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CAPN1 |
[(S)-1-((R)-1-Benzyl-2-ethylcarbamoyl-2-hydroxy-ethylcarbamoyl)-3-methyl-butyl]-carbamic acid benzyl ester |
350000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CARM1 |
5-[5-(4-Carbamimidoylphenyl)furan-2-yl]pyridine-2-carboximidamide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| CARM1 |
Furamidine |
NA |
400000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CARM1 |
PRMT5 inhibitor 4b14 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CARM1 |
Stilbamidine |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |