| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CARM1 |
1-(1-methylethyl)-N-[(6-methyl-2-oxo-4-propyl-1,2-dihydro-3-pyridinyl)methyl]-6-[6-(4-methyl-1-piperazinyl)-3-pyridinyl]-1H-indazole-4-carboxamide |
NA |
116000 |
NA |
NA |
NA |
NA |
TTD |
| CARM1 |
Gsk343 |
NA |
128000 |
NA |
NA |
NA |
NA |
TTD |
| CARM1 |
(r)-2-Amino-n-ethyl-propanamide |
NA |
105000 |
NA |
NA |
NA |
NA |
ChEMBL|TTD |
| CASP1 |
(S)-1-(4-(2-(4-methylphenylsulfonyloxy)ethoxy)benzyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP1 |
(S)-5-[1-(2-phenoxymethylpyrrolidinyl)sulfonyl]-1-(4-(tributylstannyl)benzyl)isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP1 |
2-[4-[[2,3-dioxo-5-[(2S)-2-(phenoxymethyl)pyrrolidin-1-yl]sulfonylindol-1-yl]methyl]phenoxy]ethyl 4-methylbenzenesulfonate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP1 |
(S)-1-(4-(tert-butyldimethylsilyloxy)benzyl)-5-[1-(2-phenoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP1 |
(S)-1-(4-(2-bromoethoxy)benzyl)-5-[1-(2-phenoxymethylpyrrolidinyl)sulfonyl]isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP1 |
(S)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]-1-(4-(tributylstannyl)benzyl)isatin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| CASP1 |
1-butyl-7-iodo-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP1 |
1-(3-fluoropropyl)-7-iodo-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP1 |
1-(4-fluorobutyl)-7-iodo-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP1 |
1-(4-hydroxybutyl)-7-iodo-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP1 |
7-bromo-1-(4-hydroxybutyl)-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP1 |
7-chloro-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP1 |
1-butyl-7-chloro-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP1 |
7-fluoro-5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP1 |
3-Chloro-6-(4-chloro-phenyl)-5-methyl-pyridazine-4-carboxylic acid amide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| CASP1 |
Berkchaetoazaphilone A |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP1 |
6-Chloro-[3,4'']bipyridinyl-5-carboxylic acid amide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |