Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CASP1 (S)-1-Allyl-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin NA 500000 NA NA NA NA TTD
CASP1 (S)-1-(But-3-enyl)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin NA 500000 NA NA NA NA TTD
CASP1 (S)-5-[1-(2-Methoxymethylpyrrolidinyl)sulfonyl]-1-(undec-10-enyl)isatin NA 500000 NA NA NA NA TTD
CASP1 (S)-5-[1-(2-Methoxymethylpyrrolidinyl)sulfonyl]-1-(4-vinylbenzyl)isatin NA 500000 NA NA NA NA TTD
CASP1 (S)-1-[4-(Allyloxy)benzyl]-5-[1-(2-methoxymethylpyrrolidinyl)-sulfonyl]isatin NA 500000 NA NA NA NA TTD
CASP1 6-Pyridin-4-yl-pyridazine-4-carboxylic acid amide NA 250000 NA NA NA NA TTD
CASP1 3-Methoxy-6-pyridin-4-yl-pyridazine-4-carboxylic acid amide NA 250000 NA NA NA NA TTD
CASP1 3-Chloro-6-pyridin-4-yl-pyridazine-4-carboxylic acid dimethylamide NA 250000 NA NA NA NA TTD
CASP1 3,6-dichloro-N-methylpyridazine-4-carboxamide NA 250000 NA NA NA NA TTD
CASP1 3-Methylsulfanyl-6-pyridin-4-yl-pyridazine-4-carboxylic acid amide NA 250000 NA NA NA NA TTD
CASP1 3-(2-{2-[2-Acetylamino-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-butyrylamino}-propionylamino)-propionic acid NA 200000 NA NA NA NA BindingDB
CASP1 3-Benzyloxycarbonylamino-4-oxo-9-phenyl-nonanoic acid NA|119000 1034000|NA NA NA NA NA BindingDB|TTD
CASP1 (S)-3-(benzyloxycarbonylamino)-4-oxo-5-(5-phenylpentyloxy)pentanoic acid 119000 NA NA NA NA NA BindingDB|TTD
CASP1 (S)-3-(benzyloxycarbonylamino)-5-(3-(naphthalen-1-yl)propanamidooxy)-4-oxopentanoic acid 298000 NA NA NA NA NA BindingDB|TTD
CASP1 Cannabidiol NA NA 188000 NA NA NA BindingDB
CASP1 1-Butyl-5-[2-(3-methoxypropyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione NA 500000 NA NA NA NA TTD
CASP1 1-(4-Fluorobutyl)-5-[2-(3-methoxypropyl)pyrrolidin-1-yl]sulfonylindole-2,3-dione NA 500000 NA NA NA NA TTD
CASP1 5-[(2S)-2-(ethoxymethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dione NA 500000 NA NA NA NA TTD
CASP1 5-[(2S)-2-(ethoxymethyl)pyrrolidin-1-yl]sulfonyl-1-(4-fluorobutyl)indole-2,3-dione NA 500000 NA NA NA NA TTD
CASP1 (R)-3-((S)-2-{(S)-2-[(S)-2-Acetylamino-3-(4-hydroxy-phenyl)-propionylamino]-3-methyl-butyrylamino}-propionylamino)-5-oxo-pentanoic acid NA 142000 NA NA NA NA BindingDB