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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CASP3 ethyl (2R,3R)-3-[[(1-acetylpyrrolidine-2-carbonyl)amino]-(2-amino-2-oxoethyl)carbamoyl]oxirane-2-carboxylate NA 890000 NA NA NA NA BindingDB
CASP3 Isosclerone 732120 NA NA NA NA NA BindingDB|TTD
CASP3 Pac-1 NA NA NA 113000|131000 NA NA PubChem
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-6-(4-methoxyphenyl)-2-methylpyridine-3-carboxamide NA 487200 NA NA NA NA TTD
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-6-(3-methoxyphenyl)-2-methylpyridine-3-carboxamide NA 547000 NA NA NA NA TTD
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-6-(2-methoxyphenyl)-2-methylpyridine-3-carboxamide NA 551500 NA NA NA NA TTD
CASP3 6-(3,4-dimethoxyphenyl)-N-(2-hydroxy-1-methylindol-3-yl)imino-2-methylpyridine-3-carboxamide NA 598600 NA NA NA NA TTD
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-2-methyl-6-(4-methylphenyl)pyridine-3-carboxamide NA 375300 NA NA NA NA TTD
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-2-methyl-6-(3,4,5-trimethoxyphenyl)pyridine-3-carboxamide NA 674300 NA NA NA NA TTD
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-2-methyl-6-(3-methylphenyl)pyridine-3-carboxamide NA 310000 NA NA NA NA TTD
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-2-methyl-6-(2-methylphenyl)pyridine-3-carboxamide NA 350600 NA NA NA NA TTD
CASP3 6-(4-bromophenyl)-N-(2-hydroxy-1-methylindol-3-yl)imino-2-methylpyridine-3-carboxamide NA 121700 NA NA NA NA TTD
CASP3 6-(3-bromophenyl)-N-(2-hydroxy-1-methylindol-3-yl)imino-2-methylpyridine-3-carboxamide NA 129500 NA NA NA NA TTD
CASP3 6-(2-bromophenyl)-N-(2-hydroxy-1-methylindol-3-yl)imino-2-methylpyridine-3-carboxamide NA 132400 NA NA NA NA TTD
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-2-methyl-6-phenylpyridine-3-carboxamide NA 456100 NA NA NA NA TTD
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-2-methyl-6-(4-nitrophenyl)pyridine-3-carboxamide NA 202400 NA NA NA NA TTD
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-2-methyl-6-(3-nitrophenyl)pyridine-3-carboxamide NA 278200 NA NA NA NA TTD
CASP3 N-(2-hydroxy-1-methylindol-3-yl)imino-2-methyl-6-(2-nitrophenyl)pyridine-3-carboxamide NA 296500 NA NA NA NA TTD
CASP3 2-Hydroxy-5-methylsulfamoyl-benzoic acid 1000000 NA NA NA NA NA TTD
CASP3 1-[(2,3-dioxo-1H-indol-5-yl)sulfonyl]-N-phenylpyrrolidine-2-carboxamide NA 140000 NA NA NA NA TTD