| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CASP3 |
(3S)-4-oxo-3-(pyridin-4-ylformamido)butanoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP3 |
2-(2,3-Dihydro-1,4-benzodioxin-2-yl)-1,3-thiazole-4-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP3 |
4-{[2-(2,3-Dihydro-1,4-benzodioxin-2-yl)-1,3-thiazol-4-yl]carbonyl}morpholine |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP3 |
2-(2,3-dihydro-1,4-benzodioxin-2-yl)-N,N-dimethyl-1,3-thiazole-4-carboxamide |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP3 |
2-(2,3-dihydro-1,4-benzodioxin-2-yl)-N-(furan-2-ylmethyl)-1,3-thiazole-4-carboxamide |
NA |
133000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP3 |
2-(2,3-Dihydro-1,4-benzodioxin-2-yl)-4-methyl-1,3-thiazole-5-carboxylic acid |
NA |
128000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP3 |
(2E)-3-[(4-methoxyphenyl)amino]-2-[4-(6-nitro-2-oxo-2H-chromen-3-yl)-1,3-thiazol-2-yl]prop-2-enenitrile |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CASP3 |
1-benzyl-3,7-dimethyl-8-sulfanylidene-9H-purine-2,6-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP3 |
1-ethyl-8-mercapto-3,7-dimethyl-1H-purine-2,6(3H,7H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP3 |
3-acetyl-2-(4-bromophenyl)-1-[2-(3,4-dichlorophenyl)ethyl]-4-hydroxy-2H-pyrrol-5-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CASP3 |
(S)-3-(benzyloxycarbonylamino)-5-(phenylsulfonyl)pent-4-enoic acid |
NA |
453000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP3 |
(S)-3-(benzyloxycarbonylamino)-5-(methylsulfonyl)pent-4-enoic acid |
NA |
434600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP3 |
(S)-3-(((9H-fluoren-9-yl)methoxy)carbonylamino)-5-(phenylsulfonyl)pent-4-enoic acid |
NA |
228000 |
NA |
NA |
NA |
NA |
BindingDB |
| CASP3 |
(S)-3-(((9H-fluoren-9-yl)methoxy)carbonylamino)-5-(methylsulfonyl)pent-4-enoic acid |
NA |
163200 |
NA |
NA |
NA |
NA |
BindingDB |
| CASP3 |
(S)-3-((S)-2-(benzyloxycarbonylamino)propanamido)-5-(phenylsulfonyl)pent-4-enoic acid |
NA |
343000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP3 |
(S)-3-((S)-2-(benzyloxycarbonylamino)-3-methylbutanamido)-5-(phenylsulfonyl)pent-4-enoic acid |
NA |
387900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP3 |
(S)-3-((2S,3S)-2-(benzyloxycarbonylamino)-3-methylpentanamido)-5-(phenylsulfonyl)pent-4-enoic acid |
NA |
185400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP3 |
(S)-3-((S)-2-(benzyloxycarbonylamino)propanamido)-5-(methylsulfonyl)pent-4-enoic acid |
NA |
655800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CASP3 |
(S)-3-((S)-2-(benzyloxycarbonylamino)-3-methylbutanamido)-5-(methylsulfonyl)pent-4-enoic acid |
NA |
133400 |
NA |
NA |
NA |
NA |
BindingDB |
| CASP3 |
Ac-Yvad-cho |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |