| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CD22 |
nicotinamido(-9d)NeuGc(a2-6)Gal(b)-O-Ph(4-OMe) |
NA |
132320 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CD22 |
BnNH(-9d)NeuGc(a2-6)Gal(b)-O-Ph(4-OMe) |
NA |
122570 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CD22 |
2,6-beta-D-galactopyranoside |
NA |
683330 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CD22 |
NeuGc(a2-6)Gal(b)-O-EtTMS |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CD22 |
Galf(b1-3)Gal(a1-4)3-deoxy-D-gro-D-glcNon2ulo5NAc-onic(a2-3)Gal(b1-4)Glc(b)-O-EtTMS |
NA |
NA |
2000000 |
NA |
NA |
NA |
BindingDB |
| CD274 |
6-methyl-N-(4-pyrrolidin-1-ylphenyl)pyrimidin-4-amine |
NA |
NA |
3e+06 |
NA |
NA |
NA |
ChEMBL |
| CD274 |
1-[5-(3,5-dichlorophenyl)furan-2-yl]-N-methylmethanamine |
NA |
NA |
1900000 |
NA |
NA |
NA |
ChEMBL |
| CD274 |
4-(2,3-Dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-thiazolamine |
NA |
NA |
1200000 |
NA |
NA |
NA |
ChEMBL |
| CD274 |
3-chloro-N,N-diethyl-1-benzothiophene-2-carboxamide |
NA |
NA |
2500000 |
NA |
NA |
NA |
ChEMBL |
| CD274 |
6-Methoxy-N-(3-pyridinylmethyl)-2-benzothiazolamine |
NA |
NA |
2900000 |
NA |
NA |
NA |
ChEMBL |
| CD38 |
Cyclic Inosine 5'-Diphosphoribose |
NA |
276000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CD38 |
(2R,3R,4S,5R,13R,14S,15R,16R)-18-bromo-3,4,8,10,14,15-hexahydroxy-8,10-dioxo-7,9,11,25,26-pentaoxa-1,17,19,22-tetraza-8lambda5,10lambda5-diphosphapentacyclo[18.3.1.12,5.113,16.017,21]hexacosa-18,20,22-trien-24-one |
NA |
158000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CD38 |
N'-[(Z)-(2-Hydroxyphenyl)methylidene]-2-methylfuran-3-carbohydrazide |
NA |
430000 |
NA |
NA |
NA |
NA |
TTD |
| CD38 |
N'-[(Z)-(4-Hydroxy-3-methoxyphenyl)methylidene]-2-methylfuran-3-carbohydrazide |
NA |
103000 |
NA |
NA |
NA |
NA |
TTD |
| CD38 |
N'-[(Z)-(3,4-dihydroxyphenyl)methylidene]-2-methylfuran-3-carbohydrazide |
NA |
109000 |
NA |
NA |
NA |
NA |
TTD |
| CD38 |
N'-(2-hydroxybenzoyl)-2-methylfuran-3-carbohydrazide |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CD38 |
2-Methyl-N'-[(Z)-phenylmethylidene]furan-3-carbohydrazide |
NA |
296000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CD38 |
|
NA |
103000 |
NA |
NA |
NA |
NA |
BindingDB |
| CD38 |
|
NA |
430000 |
NA |
NA |
NA |
NA |
BindingDB |
| CD38 |
|
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB |