| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CD69 |
2-[[11,23,26,28-Tetratert-butyl-17,25,27-tris(carboxymethoxy)-5-pentacyclo[19.3.1.13,7.19,13.115,19]octacosa-1(24),3,5,7(28),9,11,13(27),15(26),16,18,21(25),22-dodecaenyl]oxy]acetic acid |
NA |
251188.64 |
NA |
NA |
NA |
NA |
TTD |
| CD69 |
N-[(2R,3S,4R,5R,6R)-2-[(2R,3R,4R,5S)-4,5-dihydroxy-2-(hydroxymethyl)piperidin-3-yl]oxy-4,5-dihydroxy-6-(hydroxymethyl)oxan-3-yl]acetamide;hydrochloride |
NA |
501187.23 |
NA |
NA |
NA |
NA |
TTD |
| CD69 |
2-(Acetylamino)-2-deoxy-alpha-D-mannopyranose |
NA |
1000000000 |
NA |
NA |
NA |
NA |
TTD |
| CD69 |
2-(Acetylamino)-2-deoxy-beta-d-talopyranose |
NA |
1000000000 |
NA |
NA |
NA |
NA |
TTD |
| CDA |
2'-Deoxy-2'-methylidene-5-fluorocytidine |
25100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDA |
4-Amino-1-(3-hydroxy-5-hydroxymethyl-4-methylene-tetrahydro-furan-2-yl)-1H-pyrimidin-2-one |
1600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDA |
4-amino-1-[(4R,5R)-4-hydroxy-5-(hydroxymethyl)-3-methylideneoxolan-2-yl]pyrimidin-2-one |
7690000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDA |
1-[(3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]imidazolidin-2-one |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDA |
Cytarabine |
190000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| CDA |
1-(3,4-Dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-YL)-4-hydroxy-tetrahydro-pyrimidin-2-one |
440000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| CDC14A |
Cefsulodin |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
| CDC25A |
(N-methylpiperidino)ethanol dodecyl phosphonate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CDC25A |
2-(4-Methylmorpholin-4-ium-4-yl)ethyl tetradecyl phosphate |
NA |
290000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDC25A |
Hexadecyl 2-(1-methylpiperidinium-1-yl)ethyl phosphate |
NA |
460000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDC25A |
(N-methylpiperidino)ethanol tetradecyl phosphonate |
NA |
490000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDC25A |
Dodecyl 2-(4-methylmorpholin-4-ium-4-yl)ethyl phosphate |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDC25A |
[(4-{3-[4-(Difluoro-phosphono-methyl)-benzyloxy]-phenoxymethyl}-phenyl)-difluoro-methyl]-phosphonic acid |
NA |
163000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDC25A |
5-[3-Pyridin-2-yl-6-(5-sulfofuran-2-yl)-1,2,4-triazin-5-yl]furan-2-sulfonic acid |
NA|139000 |
110000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDC25A |
6-(2-Hydroxy-5-oxo-2,5-dihydro-furan-3-yl)-3-[(E)-4-methyl-6-(2,6,6-trimethyl-cyclohex-1-enyl)-hex-3-enyl]-5,6-dihydro-pyran-2-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDC25A |
4-[(3E,6E)-4,7-Dimethyl-9-(2,6,6-trimethyl-cyclohex-1-enyl)-nona-3,6-dienyl]-5-hydroxy-5H-furan-2-one |
NA |
990000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |