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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CDK1 2-(4-Methylmorpholin-4-ium-4-yl)ethyl tetradecyl phosphate NA 1000000 NA NA NA NA TTD
CDK1 Hexadecyl 2-(1-methylpiperidinium-1-yl)ethyl phosphate NA 1000000 NA NA NA NA TTD
CDK1 (N-methylpiperidino)ethanol tetradecyl phosphonate NA 1000000 NA NA NA NA TTD
CDK1 9H-Purin-6-amine, 9-(1-methylethyl)-N-(phenylmethyl)- NA 113000 NA NA NA NA BindingDB
CDK1 {1-[6-(3-Chloro-phenylamino)-9-isopropyl-9H-purin-2-yl]-pyrrolidin-2-yl}-methanol NA 620000 NA NA NA NA BindingDB|TTD
CDK1 Dodecyl 2-(4-methylmorpholin-4-ium-4-yl)ethyl phosphate NA 1000000 NA NA NA NA TTD
CDK1 (N-methylmorpholino)ethanol hexadecyl phosphonate NA 1000000 NA NA NA NA TTD
CDK1 4-(1H-Indol-2-Yl)Pyrimidin-2-Amine NA 140000 NA NA NA NA BindingDB
CDK1 4-(5-Bromo-1H-Indol-2-Yl)Pyrimidin-2-Amine NA 160000 NA NA NA NA BindingDB
CDK1 2-[6-(3-Chloro-phenylamino)-9-isopropyl-9H-purin-2-ylamino]-3-methyl-butan-1-ol NA 500000 NA NA NA NA BindingDB|TTD
CDK1 2-[9-Isopropyl-6-(3-trifluoromethyl-phenylamino)-9H-purin-2-ylamino]-ethanol NA 420000 NA NA NA NA BindingDB|TTD
CDK1 2-[9-Isopropyl-6-(2-trifluoromethyl-phenylamino)-9H-purin-2-ylamino]-ethanol NA 10000000 NA NA NA NA BindingDB|TTD
CDK1 2-[6-(2,4-Dichloro-phenylamino)-9-isopropyl-9H-purin-2-ylamino]-ethanol NA 2700000 NA NA NA NA BindingDB|TTD
CDK1 (2S)-2-[[6-[(4-methoxyphenyl)methylamino]-9-propan-2-ylpurin-2-yl]amino]-3-methylbutan-1-ol NA 600000 NA NA NA NA BindingDB|TTD
CDK1 2-[9-Isopropyl-6-(4-methoxy-benzylamino)-9H-purin-2-ylamino]-butan-1-ol NA 130000 NA NA NA NA BindingDB|TTD
CDK1 2-[6-(3-Chloro-phenylamino)-9-isopropyl-9H-purin-2-ylamino]-3-methyl-pentan-1-ol NA 500000 NA NA NA NA BindingDB|TTD
CDK1 2-[6-(3-Amino-4-chloro-phenylamino)-9-isopropyl-9H-purin-2-ylamino]-3-methyl-butan-1-ol NA 52000000 NA NA NA NA BindingDB|TTD
CDK1 4-[(3-Isopropyl-1H-pyrazolo[4,3-d]pyrimidin-7-ylamino)-methyl]-phenol NA 112000 NA NA NA NA BindingDB
CDK1 1-Methyl-9H-purin-6-ylamine NA 1000000 NA NA NA NA TTD
CDK1 2-Methyladenine NA 320000 NA NA NA NA BindingDB|TTD