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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CDK1 1-Amino-3-[9-isopropyl-6-(4-methoxy-benzylamino)-9H-purin-2-ylamino]-propan-2-ol NA 1600000 NA NA NA NA BindingDB|TTD
CDK1 {1-[9-Isopropyl-6-(4-methoxy-benzylamino)-9H-purin-2-ylamino]-cyclopentyl}-methanol NA 450000 NA NA NA NA BindingDB|TTD
CDK1 (2R)-1-[[6-(3-chloroanilino)-9-propan-2-ylpurin-2-yl]amino]-2,3-dihydro-1H-inden-2-ol NA 5000000 NA NA NA NA BindingDB|TTD
CDK1 2-{1-[9-Isopropyl-6-(2-phenylamino-ethylamino)-9H-purin-2-yl]-piperidin-2-yl}-ethanol NA 1500000 NA NA NA NA BindingDB|TTD
CDK1 2-[[6-(3-Chloro-phenylamino)-9-isopropyl-9H-purin-2-yl]-(4-fluoro-benzyl)-amino]-3-methyl-butan-1-ol NA 10000000 NA NA NA NA BindingDB|TTD
CDK1 2-[9-Isopropyl-6-(4-methoxy-benzylamino)-9H-purin-2-ylamino]-ethanol NA 700000 NA NA NA NA BindingDB|TTD
CDK1 2-[9-Isopropyl-6-(4-methoxy-benzylamino)-9H-purin-2-ylamino]-propane-1,3-diol NA 560000 NA NA NA NA BindingDB|TTD
CDK1 (N-methylpiperidino)ethanol 2-(hexadecyloxy)ethyl phosphonate NA 1000000 NA NA NA NA TTD
CDK1 (N-methylpiperidino)ethanol 2-(tetradecyloxy)ethyl phosphonate NA 1000000 NA NA NA NA TTD
CDK1 (N-methylmorpholino)ethanol 2-(hexadecyloxy)ethyl phosphonate NA 1000000 NA NA NA NA TTD
CDK1 (N-methylmorpholino)ethanol 2-(tetradecycloxy)ethyl phosphonate NA 1000000 NA NA NA NA TTD
CDK1 (N-methylmorpholino)ethanol 2-(dodecyloxy)ethyl phosphonate NA 1000000 NA NA NA NA TTD
CDK1 5-[(9-Isopropyl-9H-purin-6-ylamino)-methyl]-2-methoxy-phenol NA 104000 NA NA NA NA BindingDB
CDK1 2-[(9-Isopropyl-9H-purin-6-ylamino)-methyl]-phenol NA 125000 NA NA NA NA BindingDB
CDK1 (9-Isopropyl-9H-purin-6-yl)-pentyl-amine NA 144000 NA NA NA NA BindingDB
CDK1 (3-Isopropyl-1H-pyrazolo[4,3-d]pyrimidin-7-yl)-(3-methyl-but-2-enyl)-amine NA 152000 NA NA NA NA BindingDB
CDK1 Benzyl-(3-methyl-3,9-dihydro-2H-purin-6-yl)-amine NA 300000 NA NA NA NA BindingDB|TTD
CDK1 Benzyl-(1-methyl-6,9-dihydro-1H-purin-6-yl)-amine NA 1000000 NA NA NA NA TTD
CDK1 Benzyl-(7-methyl-8,9-dihydro-7H-purin-6-yl)-amine NA 1000000 NA NA NA NA TTD
CDK1 (2-Chloro-9-methyl-9H-purin-6-yl)-cyclohexyl-methyl-amine NA 130000 NA NA NA NA BindingDB|TTD