Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CDK1 | Ribociclib | NA | 113000 | NA | NA | NA | NA | BindingDB |
| CDK1 | Olomoucine | NA | 163000 | NA | NA | NA | NA | BindingDB |
| CDK1 | (2-Azepan-1-yl-9-isopropyl-9H-purin-6-yl)-(4-methoxy-benzyl)-amine | NA | 4000000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | Genistein | NA | 370000 | NA | NA | NA | NA | BindingDB|PubChem |
| CDK1 | 9-Bromo-5-ethylpaullone | NA | 470000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | 9-Bromo-5,7,12-tri-(tert-butyloxycarbonyl)-paullone | NA | 150000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | 9-Bromo-5,12-bis-(tert-butyloxycarbonyl)-paullone | NA | 1000000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | N6-Benzyladenine | NA | 200000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | 3-Methyl-3,9-dihydro-2H-purin-6-ylamine | NA | 400000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | 6-Chloro-2-iodo-9-isopropyl-9H-purine | NA | 150000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | 2,6,9-Trisubstituted purine deriv. 6 | NA | 470000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | 2,6,9-Trisubstituted purine deriv. 7 | NA | 150000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | 2,6,9-Trisubstituted purine deriv. 8 | NA | 110000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | 2,6,9-Trisubstituted purine deriv. 25 | NA | 200000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | Cvt-313 | NA | 330000 | NA | NA | NA | NA | BindingDB|TTD |
| CDK1 | 9-Methyladenine | NA | 350000 | NA | NA | NA | NA | TTD |
| CDK1 | N-(5,6-Diphenylfuro[2,3-D]pyrimidin-4-YL)glycine | NA | 200000 | NA | NA | NA | NA | TTD |
| CDK1 | 2-Chloroadenine | NA | 1000000 | NA | NA | NA | NA | TTD |
| CDK1 | 10-Chloro-6-hydroxy-11lambda5-pyrido(1,2-A)quinolin-11-ylium chloride | NA | 1000000 | NA | NA | NA | NA | TTD |
| CDK1 | 2-[9-Isopropyl-6-(4-methoxy-benzylamino)-9H-purin-2-ylamino]-1-phenyl-ethanol | NA | 2800000 | NA | NA | NA | NA | BindingDB|TTD |