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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CDK2 (S)-{1-[2-(2-chlorophenyl)-5-hydroxy-4-oxo-4H-chromen-8-ylcarbamoyl]-2-phenylethyl}carbamic acid tert-butyl ester NA 417000 NA NA NA NA BindingDB
CDK2 (S)-{1-[2-(2-chlorophenyl)-5-hydroxy-4-oxo-4H-chromen-8-ylcarbamoyl]-3-methylbutyl}carbamic acid tert-butyl ester NA 417000 NA NA NA NA BindingDB
CDK2 sec-butyl 2-(2-chlorophenyl)-5-hydroxy-4-oxo-4H-chromen-8-ylcarbamate NA 417000 NA NA NA NA BindingDB
CDK2 N-[2-(2-chlorophenyl)-5-hydroxy-4-oxo-4H-chromen-8-yl]benzenesulfonamide NA 178000 NA NA NA NA BindingDB
CDK2 4-chloro-N-[2-(2-chlorophenyl)-5,7-dihydroxy-4-oxo-4H-chromen-8-yl]benzamide NA 339000 NA NA NA NA BindingDB
CDK2 2-(2-Chlorophenyl)-5-hydroxy-8-pyrrolidin-1-ylchromen-4-one NA 417000 NA NA NA NA BindingDB
CDK2 NA 109000 NA NA NA NA BindingDB
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-4''-fluoro-N-methylbiphenyl-4-carboxamide NA 875000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-4''-tert-butyl-N-methylbiphenyl-4-carboxamide NA 745000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-4''-methoxy-N-methylbiphenyl-4-carboxamide NA 289000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-4''-fluorobiphenyl-4-carboxamide NA 764000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-4''-methylbiphenyl-4-carboxamide NA 816000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-4''-tert-butylbiphenyl-4-carboxamide NA 790000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-4''-methoxybiphenyl-4-carboxamide NA 1085000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)biphenyl-3-carboxamide NA 1002000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-4''-fluorobiphenyl-2-carboxamide NA 1216000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-4''-tert-butylbiphenyl-2-carboxamide NA 262000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-4''-methoxybiphenyl-2-carboxamide NA 921000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-3''-methoxybiphenyl-2-carboxamide NA 926000 NA NA NA NA BindingDB|TTD
CDK2 N-(2-(1H-Indol-3-yl)ethyl)-2''-methoxybiphenyl-2-carboxamide NA 375000 NA NA NA NA BindingDB|TTD