| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CDK2 |
N-(2-(1H-Indol-3-yl)ethyl)-3''-fluorobiphenyl-2-carboxamide |
NA |
417000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4''-fluorobiphenyl-2-yl)methanone |
NA |
357000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3''-fluorobiphenyl-2-yl)methanone |
NA |
480000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2''-fluorobiphenyl-2-yl)methanone |
NA |
434000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
[2-(3-Methylphenyl)phenyl]-(1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl)methanone |
NA |
386000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
[3-(4-Fluorophenyl)phenyl]-(1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl)methanone |
NA |
318000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3''-fluorobiphenyl-3-yl)methanone |
NA |
611000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2''-fluorobiphenyl-3-yl)methanone |
NA |
335000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4''-methylbiphenyl-3-yl)methanone |
NA |
466000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3''-methylbiphenyl-3-yl)methanon |
NA |
465000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2''-methylbiphenyl-3-yl)methanone |
NA |
665000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3''-methoxybiphenyl-3-yl)methanone |
NA |
362000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
Biphenyl-3-yl(3,4-dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)methanone |
NA |
1109000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4''-fluorobiphenyl-4-yl)methanone |
NA |
438000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3''-fluorobiphenyl-4-yl)methanone |
NA |
296000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2''-fluorobiphenyl-4-yl)methanone |
NA |
310000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3''-methylbiphenyl-4-yl)methanone |
NA |
405000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2''-methylbiphenyl-4-yl)methanone |
NA |
340000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3''-methoxybiphenyl-4-yl)methanone |
NA |
424000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CDK2 |
(3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2''-methoxybiphenyl-4-yl)methanone |
NA |
321000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |