| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CHKA |
|
NA |
NA |
340000 |
NA |
NA |
NA |
BindingDB |
| CHKA |
|
NA |
NA |
630000 |
NA |
NA |
NA |
BindingDB |
| CHKA |
|
NA |
NA |
194000 |
NA |
NA |
NA |
BindingDB |
| CHRFAM7A |
Acetylcholine |
NA |
NA |
NA |
155000|230000|180000 |
NA |
NA |
PubChem |
| CHRFAM7A |
Imidacloprid |
NA |
270000 |
NA |
NA |
NA |
NA |
PubChem |
| CHRFAM7A |
Nicotine |
NA |
NA |
NA |
113000 |
NA |
NA |
PubChem |
| CHRM1 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
259998 |
PubChem |
| CHRM1 |
rac-N,N-dimethyl-2-(3-(1-(thiazol-2-yl)ethyl)benzo[b]thiophen-2-yl)ethanamine |
2072000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CHRM1 |
Moxifloxacin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRM1 |
(-)-(S)-9-Fluoro-2,3-dihydro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-7H-pyrido(1,2,3-de)-1,4-benzoxazine-6-carboxylic acid, hemihydrate |
NA |
NA |
NA |
NA |
NA |
300000|140001 |
PubChem |
| CHRM1 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRM1 |
2-(Furan-2-yl)pyrrolidine |
177827.94 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CHRM1 |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRM1 |
Ofloxacin |
NA |
NA |
NA |
NA |
NA |
189998|300000 |
PubChem |
| CHRM1 |
(-)-(R)-2-(3-(1-(1H-pyrazol-1-yl)ethyl)benzo[b]thiophen-2-yl)-N,N-dimethylethanamine |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CHRM1 |
(-)-(R)-N,N-dimethyl-2-(3-(1-(thiazol-4-yl)ethyl)benzo[b]thiophen-2-yl)ethanamine |
4759000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CHRM1 |
(-)-(R)-N,N-dimethyl-2-(3-(1-(thiazol-5-yl)ethyl)benzo[b]thiophen-2-yl)ethanamine |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CHRM1 |
5-[[(E)-1-azabicyclo[2.2.2]octan-3-ylmethylideneamino]oxymethyl]-1,2-oxazole-3-carbonitrile;hydrochloride |
NA |
132700 |
NA |
NA |
NA |
NA |
TTD |
| CHRM1 |
N-cyclohexyl-2-(4-methyl-1,4-diazepan-1-yl)acetamide |
NA |
102000 |
NA |
NA |
NA |
NA |
TTD |
| CHRM1 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |