| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CHRM2 |
(2S)-2-(furan-2-yl)pyrrolidine |
107151.93 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CHRM2 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRM3 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRM3 |
N-[2-(dimethylamino)ethyl]-3-(pyridin-4-ylmethyl)-1H-indene-2-carboxamide |
134896|134896.29 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CHRM3 |
4-[Hydroxy(diphenyl)methyl]-1-(2-hydroxyethyl)-1-azoniabicyclo[2.2.2]octane Bromide |
NA |
486000 |
NA |
NA |
NA |
NA |
TTD |
| CHRM3 |
Umeclidinium metabolite M14 |
NA |
486000 |
NA |
NA |
NA |
NA |
BindingDB |
| CHRM3 |
4-[Hydroxy(diphenyl)methyl]-1-propyl-1-azoniabicyclo[2.2.2]octane bromide |
NA |
208000 |
NA |
NA |
NA |
NA |
TTD |
| CHRM3 |
4-[Hydroxy(diphenyl)methyl]-1-propyl-1-azoniabicyclo[2.2.2]-octane Bromide |
NA |
208000 |
NA |
NA |
NA |
NA |
BindingDB |
| CHRM3 |
1-Butyl-4-[hydroxy(diphenyl)methyl]-1-azoniabicyclo[2.2.2]octane bromide |
NA |
135000 |
NA |
NA |
NA |
NA |
TTD |
| CHRM3 |
1-Butyl-4-[hydroxy(diphenyl)methyl]-1-azoniabicyclo[2.2.2]-octane Bromide |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB |
| CHRM3 |
1-Ethyl-4-[hydroxy(diphenyl)methyl]-1-azoniabicyclo[2.2.2]octane bromide |
NA |
104000 |
NA |
NA |
NA |
NA |
TTD |
| CHRM3 |
1-Ethyl-4-[hydroxy(diphenyl)methyl]-1-azoniabicyclo[2.2.2]-octane Bromide |
NA |
104000 |
NA |
NA |
NA |
NA |
BindingDB |
| CHRM3 |
Moxifloxacin |
NA |
NA |
NA |
NA |
NA |
219999 |
PubChem |
| CHRM3 |
3-(3-Amino-1,2,4-oxadiazol-5-yl)-1-azabicyclo(2.2.1)heptane |
NA |
NA |
NA |
104000 |
NA |
NA |
BindingDB|TTD |
| CHRM3 |
Ethyl 4-(2-(2-methylbenzamido)ethylamino)piperidine-1-carboxylate |
NA|189600 |
NA |
NA |
360100|NA |
NA |
NA |
BindingDB |
| CHRM3 |
(-)-(S)-9-Fluoro-2,3-dihydro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-7H-pyrido(1,2,3-de)-1,4-benzoxazine-6-carboxylic acid, hemihydrate |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRM3 |
3-Quinuclidinemethanol, alpha,alpha-diphenyl-, hydrobromide |
NA |
1104000 |
NA |
NA |
NA |
NA |
TTD |
| CHRM3 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRM3 |
4-(Hydroxydiphenylmethyl)-1-azoniabicyclo[2.2.2]octane bromide |
NA |
1068000 |
NA |
NA |
NA |
NA |
BindingDB |
| CHRM3 |
Diphenyl-[1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octan-3-yl]methanol;bromide |
NA |
2824000 |
NA |
NA |
NA |
NA |
TTD |