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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CHRM3 3-[Hydroxy(diphenyl)methyl]-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane Bromide NA 2824000 NA NA NA NA BindingDB
CHRM3 1,1-Diphenyl-2-[1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octan-3-yl]ethanol;bromide NA 122000 NA NA NA NA TTD
CHRM3 3-(2-Hydroxy-2,2-diphenylethyl)-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane Bromide NA 122000 NA NA NA NA BindingDB
CHRM3 4-[Hydroxy(diphenyl)methyl]-1-methyl-1-azoniabicyclo[2.2.2]octane bromide NA 935000 NA NA NA NA TTD
CHRM3 4-[Hydroxy(diphenyl)methyl]-1-methyl-1-azoniabicyclo[2.2.2]-octane Bromide NA 935000 NA NA NA NA BindingDB
CHRM3 1-(Cyclopropylmethyl)-4-[hydroxy(diphenyl)methyl]-1-azoniabicyclo[2.2.2]octane Bromide NA 1956000 NA NA NA NA TTD
CHRM3 [1-(Cyclopropylmethyl)-1-azoniabicyclo[2.2.2]octan-4-yl]-diphenylmethanol NA 1956000 NA NA NA NA BindingDB
CHRM3 [1-(2-Aminoethyl)-1-azoniabicyclo[2.2.2]octan-4-yl]-diphenylmethanol;bromide NA 850000 NA NA NA NA TTD
CHRM3 [1-(2-Aminoethyl)-1-azoniabicyclo[2.2.2]oct-4-yl](diphenyl)-methanolate bromide NA 850000 NA NA NA NA BindingDB
CHRM3 3-[4-[Hydroxy(diphenyl)methyl]-1-azoniabicyclo[2.2.2]octan-1-yl]propan-1-ol;bromide NA 29509000 NA NA NA NA TTD
CHRM3 4-[Hydroxy(diphenyl)methyl]-1-(3-hydroxypropyl)-1-azoniabicyclo[2.2.2]octane Bromide NA 29509000 NA NA NA NA BindingDB
CHRM3 4-[Hydroxy(diphenyl)methyl]-1-[3-(methyloxy)propyl]-1-azoniabicyclo[2.2.2]octane Bromide NA 829000 NA NA NA NA TTD
CHRM3 [1-(3-Methoxypropyl)-1-azoniabicyclo[2.2.2]octan-4-yl]-diphenylmethanol NA 829000 NA NA NA NA BindingDB
CHRM3 [1-(5-Phenoxypentyl)-1-azoniabicyclo[2.2.2]octan-4-yl]-diphenylmethanol;bromide NA 306000 NA NA NA NA TTD
CHRM3 4-[Hydroxy(diphenyl)methyl]-1-[5-(phenyloxy)pentyl]-1-azoniabicyclo[2.2.2]octane Bromide NA 306000 NA NA NA NA BindingDB
CHRM3 2-[2-[4-[Hydroxy(diphenyl)methyl]-1-azoniabicyclo[2.2.2]octan-1-yl]ethoxymethyl]benzonitrile;bromide NA 5403000 NA NA NA NA TTD
CHRM3 1-(2-{[(2-Cyanophenyl)methyl]oxy}ethyl)-4-[hydroxy(diphenyl)methyl]-1-azoniabicyclo[2.2.2]octane Bromide NA 5403000 NA NA NA NA BindingDB
CHRM3 Meropenem NA NA NA NA NA 300000 PubChem
CHRM3 N-chloromethyl-brucine NA NA 501187 NA NA NA GtoPDB
CHRM3 Ofloxacin NA NA NA NA NA 300000 PubChem