| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CSGALNACT1 |
(2S)-2-[[5-[4-[(4-chloro-2-phenoxyphenyl)carbamoylamino]phenyl]-1,3-oxazole-2-carbonyl]amino]-3-methylbutanoic acid |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSGALNACT1 |
(2S)-2-[[3-[4-[(2,4-difluorophenyl)carbamoylamino]phenyl]-1,2,4-oxadiazole-5-carbonyl]amino]-3-methylbutanoic acid |
NA |
259000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSGALNACT1 |
(2S)-2-[[3-[4-[(2-fluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid |
NA |
141000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSGALNACT1 |
(2S)-2-[[3-[4-[(2,5-difluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid |
NA |
141000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSGALNACT1 |
(2S)-2-[[3-[4-[(2,6-difluorophenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid |
NA |
185000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSGALNACT1 |
(2S)-2-[[3-[4-[(3,5-dimethylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSGALNACT1 |
(2S)-2-[[3-[4-[(3-fluoro-4-methylphenyl)carbamoylamino]phenyl]-1,2-oxazole-5-carbonyl]amino]-3-methylbutanoic acid |
NA |
178000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSK |
(S)-N-hydroxy-3-(4-hydroxyphenyl)-2-phenylpropanamide |
NA |
290000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CSK |
(S)-2-amino-N-benzyl-N-hydroxy-3-(4-hydroxyphenyl)propanamide |
NA |
291000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CSNK1A1 |
N-(2-aminoethyl)isoquinoline-5-sulfonamide |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSNK1A1 |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CSNK1A1 |
4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diol |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CSNK1A1 |
Rki-1447 |
NA |
469800 |
NA |
NA |
NA |
NA |
BindingDB |
| CSNK1A1 |
1-[(3-Hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea;methanesulfonic acid |
NA |
469800 |
NA |
NA |
NA |
NA |
TTD |
| CSNK1D |
6-(1,9-Diazaspiro[5.5]undecan-9-Yl)-9h-Purine |
NA |
238000 |
NA |
NA |
NA |
NA |
TTD |
| CSNK1E |
AR-AO-14418 |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| CSNK1E |
1-[(4-methoxyphenyl)methyl]-3-[6-(2H-tetrazol-5-yl)-1,3-benzothiazol-2-yl]urea |
NA |
15300000 |
NA |
NA |
NA |
NA |
TTD |
| CSNK1E |
1-[(4-methoxyphenyl)methyl]-3-[4-(2H-tetrazol-5-yl)pyridin-2-yl]urea |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| CSNK1E |
1-[(4-Methoxyphenyl)methyl]-3-(6-nitro-1,3-benzothiazol-2-yl)urea |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| CSNK1E |
1-(4-Cyanopyridin-2-yl)-3-[(4-methoxyphenyl)methyl]urea |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |