Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CRBN | 2-Piperidone | 146000 | NA | NA | NA | NA | NA | BindingDB |
| CRBN | 2-amino-N-(2,6-dioxopiperidin-3-yl)-6-fluorobenzamide | NA | 114000 | NA | NA | NA | NA | BindingDB |
| CRBN | 2-acetamido-N-(2,6-dioxopiperidin-3-yl)thiophene-3-carboxamide | NA | 131000 | NA | NA | NA | NA | BindingDB |
| CRBN | N-(2,6-Dioxo-3-piperidinyl)benzamide | NA | 127000 | NA | NA | NA | NA | BindingDB |
| CRBN | Sofosbuvir | NA | 1000000 | NA | NA | NA | NA | PubChem |
| CRBN | Rolipram | 102000|NA | NA|202000 | NA | NA | NA | NA | PubChem |
| CRBN | Uridine | 390000|NA | NA|757000 | NA | NA | NA | NA | PubChem |
| CRBN | Uridine Monophosphate | NA | 5000000 | NA | NA | NA | NA | PubChem |
| CRBN | Dimethyl Sulfone | NA|137490000 | 181000000|NA | NA | NA | NA | NA | PubChem|TTD |
| CRBN | N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide | NA | 133000 | NA | NA | NA | NA | BindingDB |
| CRBN | 3-amino-N-(2,6-dioxopiperidin-3-yl)benzamide | NA | 107000 | NA | NA | NA | NA | BindingDB |
| CRBN | 4-amino-N-(2,6-dioxopiperidin-3-yl)-2-methylbenzamide | NA | 132000 | NA | NA | NA | NA | BindingDB |
| CRBN | Dimethyl Sulfoxide | NA|137000|137000000 | 264000|NA | NA | NA | NA | NA | PubChem |
| CRBN | Furagin | NA | 1000000 | NA | NA | NA | NA | PubChem |
| CRBN | Glutarimide | 103100 | NA | NA | NA | NA | NA | TTD |
| CREBBP | Butyrolactone 3 | NA | 500000 | NA | NA | NA | NA | TTD |
| CREBBP | (2R)-2-ethyl-1,2,3,5-tetrahydro-1,5-benzodiazepin-4-one | NA | 120000 | NA | NA | NA | NA | BindingDB|ChEMBL|TTD |
| CREBBP | 4,4-dimethyl-2,3,4,5-tetrahydro-1H-1,5-benzodiazepin-2-one | NA | 200000 | NA | NA | NA | NA | TTD |
| CREBBP | Methyl 2-oxo-2,3-dihydro-1,3-benzoxazole-6-carboxylate | NA | 455000 | NA | NA | NA | NA | BindingDB|ChEMBL|TTD |
| CREBBP | (2R,3R)-4-methylidene-5-oxo-3-propyloxolane-2-carboxylic acid | NA | 500000 | NA | NA | NA | NA | BindingDB|TTD |