| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CPT1B |
4-Hydroxyphenylglyoxylic acid |
NA |
510000 |
NA |
NA |
NA |
NA |
BindingDB |
| CPT2 |
(S)-2-Hexadecyl-2-hydroxy-4,4-dimethyl-morpholin-4-ium; bromide |
NA |
235000 |
NA |
NA |
NA |
NA |
BindingDB |
| CRAT |
3-Amino-5,5-dimethylhexanoic acid |
2600000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CRAT |
3-Acetamido-5,5-dimethylhexanoic acid |
25000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CRAT |
(S)-3-Amino-5,5-dimethylhexanoic acid |
1900000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CRAT |
(3r)-3-Hydroxy-5,5-Dimethylhexanoic Acid |
7500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CRAT |
(3S)-3-hydroxy-5,5-dimethylhexanoic acid |
20300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CRAT |
3-Hydroxy-5,5-dimethylhexanoic acid |
8300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CRAT |
3-Amino-5,5-dimethyl-hexanoic acid anion |
2600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CRAT |
(R)-3-Hydroxy-5,5-dimethyl-hexanoic acid anion |
7500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CRAT |
(S)-3-Hydroxy-5,5-dimethyl-hexanoic acid anion |
20300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CRAT |
3-Acetyl-5,5-dimethyl-hexanoic acid anion |
4100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CRAT |
3-Acetyl-5,5-dimethylhexanoic acid |
4100000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CRAT |
(S)-3-Amino-5,5-dimethyl-hexanoic acid anion |
1900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CRAT |
3-Hydroxy-5,5-dimethyl-hexanoic acid anion |
8300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CRAT |
3-Acetylamino-5,5-dimethyl-hexanoic acid anion |
25000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CRAT |
(R)-3-Amino-5,5-dimethyl-hexanoic acid anion |
9200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CRAT |
(3R)-3-amino-5,5-dimethylhexanoic acid |
9200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CRAT |
3-Amino-4-(trimethylazaniumyl)butanoate |
4000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CRBN |
Uracil |
NA|212000 |
415000|NA |
NA |
NA |
NA |
NA |
PubChem |