| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CPB1 |
2-(4-benzyl-5-(3-methylphenethyl)-4H-1,2,4-triazol-3-ylthio)acetic acid |
196000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CPB1 |
N-(2-(2-(2-(4-methoxyphenyl)-2-oxoethyl)-2H-tetrazol-5-yl)phenyl)cyclopropanecarboxamide |
292000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CPB2 |
2-[(6-Amino-5-chloropyridin-3-yl)methyl]-3-propanoylselanylpropanoic acid |
NA |
370000 |
NA |
NA |
NA |
NA |
BindingDB |
| CPB2 |
2-Amino-3-(1-aminoisoquinolin-7-yl)propanoic acid, 2 |
145000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CPB2 |
2-Amino-3-(1-aminoisoquinolin-6-yl)propanoic acid, 1 |
220000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CPB2 |
Ethyl 2-[(6-aminopyridin-3-yl)methyl]-3-propanoylselanylpropanoate |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CPB2 |
Ethyl 2-(acetylsulfanylmethyl)-7-aminoheptanoate |
NA |
310000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CPN1 |
(3S)-3-(4-aminobutyl)-1-[[4-fluoro-2-(3-methylimidazol-4-yl)phenyl]methyl]-4-hydroxy-4-oxo-1,4lambda5-azaphosphinane-3-carboxylic acid |
282000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| CPN1 |
2-[(6-Amino-5-chloropyridin-3-yl)methyl]-3-propanoylselanylpropanoic acid |
NA |
380000 |
NA |
NA |
NA |
NA |
TTD |
| CPN1 |
(5r)-5-(3-Aminopropyl)-1-Propyl-4,5,6,7-Tetrahydro-1h-Benzimidazole-5-Carboxylic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CPN1 |
(5R)-5-(3-aminopropyl)-1-(3-methylbutyl)-6,7-dihydro-4H-benzimidazole-5-carboxylic acid;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CPN1 |
(5R)-5-(3-aminopropyl)-1-cyclohexyl-6,7-dihydro-4H-benzimidazole-5-carboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CPN1 |
(5R)-5-(3-aminopropyl)-1-[(3-phenylphenyl)methyl]-6,7-dihydro-4H-benzimidazole-5-carboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CPN1 |
5-(3-aminopropyl)-1-[2-(4-cyclohexylcyclohexyl)ethyl]-6,7-dihydro-4H-benzimidazole-5-carboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CPN1 |
5-(3-aminopropyl)-1-phenyl-6,7-dihydro-4H-benzimidazole-5-carboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CPN1 |
7-(3-aminopropyl)-3-ethyl-6,8-dihydro-5H-imidazo[1,2-a]pyridine-7-carboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CPN1 |
(7R)-7-(3-aminopropyl)-3-phenyl-6,8-dihydro-5H-imidazo[1,2-a]pyridine-7-carboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CPN1 |
(7R)-7-(3-aminopropyl)-3-[3-(2,4-dichlorophenyl)phenyl]-6,8-dihydro-5H-imidazo[1,2-a]pyridine-7-carboxylic acid;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CPT1A |
Amiodarone |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| CPT1A |
2,6-Ditert-butyl-4-[3-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]propylsulfanyl]phenol |
NA |
16800000|51000000 |
NA |
NA |
NA |
NA |
BindingDB |