| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CNR1 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CNR1 |
Example 133 in WO2010036630 |
NA |
NA |
NA |
200000 |
NA |
NA |
BindingDB |
| CNR1 |
N-[2-(4-fluorophenyl)ethyl]-8-hydroxy-7-methoxy-1-methyl-2-oxo-6-pentylquinoline-3-carboxamide |
864000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CNR1 |
N-[2-(4-fluorophenyl)ethyl]-8-hydroxy-7-methoxy-2-oxo-6-pentyl-1H-quinoline-3-carboxamide |
2398000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CNR1 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| CNR1 |
4-[[2-(Oxan-4-ylmethylcarbamoyl)pyridin-3-yl]carbamoyl]naphthalene-1-carboxylic acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| CNR1 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| CNR1 |
2-[2-Methyl-6-(4-methyl-piperazin-1-yl)-9-(tetrahydro-pyran-4-yl)-9h-purin-8-yl]-benzonitrile hydrochloride salt |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CNR1 |
(4-Fluoronaphthalen-1-yl)-(2-methyl-1-propylindol-3-yl)methanone |
NA |
NA |
NA |
268000 |
NA |
NA |
BindingDB |
| CNR1 |
N-(cyclobutylmethyl)-3-[[4-(methylsulfonylmethyl)naphthalene-1-carbonyl]amino]pyridine-2-carboxamide |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| CNR1 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CNR1 |
US10570125, Example 1 |
NA |
NA|104000 |
NA |
104000|NA |
NA |
NA |
BindingDB |
| CNR1 |
US10112934, Example 2 |
NA |
NA |
NA |
150000|200000 |
NA |
NA |
BindingDB |
| CNR1 |
US10112934, Example 3 |
NA |
NA |
NA |
200000 |
NA |
NA |
BindingDB |
| CNR1 |
US10112934, Example 7 |
NA |
NA |
NA |
200000 |
NA |
NA |
BindingDB |
| CNR2 |
N-cyclohexyl-1-(2,4-dichlorophenyl)-6-methyl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide |
131825673.9 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CNR2 |
MK-3168 |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| CNR2 |
6-bromo-N-hexyl-4-oxo-1-pentylquinoline-3-carboxamide |
1122018.45 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CNR2 |
(6AR,10AR)-3-(1,1-Dimethylbutyl)-6A,7,10,10A-tetrahydro-6,6,9-trimethyl-6H-dibenzo[B,D]pyran |
NA |
NA |
NA |
168600 |
NA |
NA |
BindingDB |
| CNR2 |
Epigallocatechin |
361300 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |