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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CMA1 Vaborbactam NA 1000000 NA NA NA NA PubChem|TTD
CMA1 Tetrahydroisoquinoline hydantoin derivative, 4c NA 308000 NA NA NA NA BindingDB
CMA1 Tetrahydroisoquinoline hydantoin derivative, 4d NA 123000 NA NA NA NA BindingDB
CMA1 6-Chloro-1,3-dihydroindol-2-one NA 470000 NA NA NA NA BindingDB|ChEMBL|TTD
CMA1 6-Chloroindole NA 340000 NA NA NA NA BindingDB|ChEMBL|TTD
CMA1 Tetrahydroisoquinoline hydantoin derivative, 3a NA 171500 NA NA NA NA BindingDB
CMA1 Tetrahydroisoquinoline hydantoin derivative, 3b NA 205500 NA NA NA NA BindingDB
CMA1 Tetrahydroisoquinoline hydantoin derivative, 3c NA 373500 NA NA NA NA BindingDB
CNR1 Imipenem NA NA NA NA NA 300000 PubChem
CNR1 US10112934, Example 1 NA NA NA 104000 NA NA BindingDB
CNR1 N-[2-(4-fluorophenyl)ethyl]-7-methoxy-2-oxo-8-propoxy-1H-quinoline-3-carboxamide 336000 NA NA NA NA NA BindingDB|TTD
CNR1 N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(4-chlorophenylsulfonyl)-2-methylpropanamide NA NA NA 700000 NA NA BindingDB
CNR1 N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-(4-chlorophenylsulfonyl)-2-methylpropanamide NA NA NA 223000 NA NA BindingDB
CNR1 SR 144528 NA|116800 541900|NA NA NA NA NA BindingDB
CNR1 Cefazolin NA NA NA NA NA 300000 PubChem
CNR1 Meropenem NA NA NA NA NA 300000 PubChem
CNR1 N-[3-(2-hydroxy-1,1-dimethyl-ethyl)-isoxazol-5-yl]-2-methyl-2-(tetrahydro-pyran-4-sulfonyl)-propionamide NA NA|150000 NA 150000|NA NA NA BindingDB
CNR1 Example 30 in WO2010147792 NA NA|120000 NA 120000|NA NA NA BindingDB
CNR1 (E)-2-(benzenesulfonyl)-3-[1-(2-piperidin-1-ylethyl)indol-3-yl]prop-2-enenitrile 163400 NA NA NA NA NA BindingDB|TTD
CNR1 Cefepime NA NA NA NA NA 300000 PubChem