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negative DTIs
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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
CISD1
4-Chloro-5-sulfamoyl-2-(undecylamino)benzoic acid
NA
190000
NA
NA
NA
NA
BindingDB
CISD1
4-Chloro-2-(dodecylamino)-5-sulfamoylbenzoic acid
NA
NA
NA
236400
NA
NA
BindingDB
CISD1
4-Chloro-2-[(4-chlorophenyl)methylamino]-5-sulfamoylbenzoic acid
NA
NA
NA
100580
NA
NA
BindingDB
CISD1
4-Amino-1,8-naphthalimide
NA
264000
NA
NA
NA
NA
BindingDB
CISD1
Furosemide [USAN:USP:INN:BAN:JAN]
NA
101900
NA
NA
NA
NA
BindingDB|PubChem
CISD1
Gemfibrozil
NA
170600
NA
NA
NA
NA
BindingDB|PubChem
CISD1
2-Amino-5-benzyl-1,3-thiazol-4-ol
NA
37320000
NA
NA
NA
NA
BindingDB
CKM
3-(1-Amino-2-phosphonatoethylidene)azaniumylpropanoate
37000000
NA
NA
NA
NA
NA
BindingDB
CKM
2-[(1-Amino-2-phosphonatoethylidene)-methylazaniumyl]acetate
1400000
NA
NA
NA
NA
NA
BindingDB
CKM
2-(1-Amino-2-phosphonatoethylidene)azaniumylacetate
5700000
NA
NA
NA
NA
NA
BindingDB
CLCN6
4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid
NA
1000000
NA
NA
NA
NA
GtoPDB
CLCN7
5-Nitro-2-(3-phenylpropylamino)benzoic acid
NA
156000
NA
NA
NA
NA
GtoPDB
CLEC4C
4'-(alpha-D-Mannopyranosyloxy)-biphenyl-4-carboxylic acid
NA
1000000
NA
NA
NA
NA
BindingDB
CLEC4M
N-Acetyl-D-Mannosamine
NA
6900000
NA
NA
NA
NA
PubChem
CLEC4M
Niflumic Acid
NA
610000
NA
NA
NA
NA
PubChem
CLK1
N,5-bis(4-hydroxyphenyl)-1H-pyrrolo[2,3-b]pyridine-3-carboxamide
NA
NA
NA
1000000
NA
NA
TTD
CLK1
4-[3-(4-hydroxyphenyl)-1H-indazol-5-yl]phenol
NA
NA
NA
1000000
NA
NA
TTD
CLK1
4-[3-(1H-indol-5-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenol
NA
NA
NA
117000
NA
NA
BindingDB|TTD
CLK1
4-[5-(4-nitrophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]phenol
NA
NA
NA
187000
NA
NA
BindingDB|TTD
CLK1
4-[3-(4-aminophenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenol
NA
NA
NA
1000000
NA
NA
TTD
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