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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
CHRNB4
[1-[3-(4-Phenyltriazol-1-yl)propyl]piperidin-3-yl]methyl 2-phenylbenzoate
NA
389045.14
NA
NA
NA
NA
TTD
CHRNB4
[1-(3-Phenylpropanoyl)piperidin-3-yl]methyl 2-phenylbenzoate
NA
331131.12
NA
NA
NA
NA
TTD
CHRNB4
2-phenyl-N-[[1-(3-phenylpropyl)piperidin-3-yl]methyl]benzamide
NA
100000000
NA
NA
NA
NA
TTD
CHRNE
(2E)-6-methoxy-2-[[4-(1-quinolin-4-yltriazol-4-yl)phenyl]methylidene]-3H-inden-1-one
NA
104000
NA
NA
NA
NA
BindingDB
CHRNE
(2E)-5-methoxy-2-[[4-(1-quinolin-4-yltriazol-4-yl)phenyl]methylidene]-3H-inden-1-one
NA
114000
NA
NA
NA
NA
BindingDB
CHRNE
1-[(3,5-Diphenyl-1,2,4-triazole-1-carbonyl)amino]-3-methylurea
NA
1600000
NA
NA
NA
NA
BindingDB
CHRNE
1-[(4-Bromophenyl)methyl]-3,5-diphenyl-1,2,4-triazole
NA
1560000
NA
NA
NA
NA
BindingDB
CHURC1-FNTB
Lonafarnib
NA
500000
NA
NA
NA
NA
PubChem
CHURC1-FNTB
Ethylenediamine
NA
15500000
NA
NA
NA
NA
PubChem
CIB1
Bufotenin
NA
NA
NA
NA
112202
NA
PubChem
CIB1
Oxyquinoline
NA
NA
NA
NA
125892
NA
PubChem
CIB1
Glutamic Acid
NA
NA
NA
NA
112202
NA
PubChem
CIB1
Malathion
NA
NA
NA
NA
112202
NA
PubChem
CIB1
Psilocin
NA
NA
NA
NA
125892
NA
PubChem
CIB1
Nitrofurazone
NA
NA
NA
NA
112202
NA
PubChem
CIB1
Thiotepa
NA
NA
NA
NA
125892
NA
PubChem
CIB1
Trazodone
NA
NA
NA
NA
112202
NA
PubChem
CIB1
Verapamil Hydrochloride
NA
NA
NA
NA
112202
NA
PubChem
CISD1
(Z)-5-Benzylidene-2-iminothiazolidin-4-one
NA|1594000
37320000|NA
NA
NA
NA
NA
BindingDB
CISD1
4-Chloro-2-[(4-phenylphenyl)methylamino]-5-sulfamoylbenzoic acid
NA
NA
NA
106700
NA
NA
BindingDB
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