| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CLK1 |
N-(3-hydroxyphenyl)-5-(4-hydroxyphenyl)-1H-pyrrolo[2,3-b]pyridine-3-carboxamide |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CLK1 |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CLK1 |
4-[3-(4-hydroxyphenyl)-1H-indol-5-yl]phenol |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CLPP |
hClpP-activator-D9 |
NA |
NA |
NA |
110000 |
NA |
NA |
BindingDB |
| CLTC |
6-Amino-1,3-dioxo-2-propylbenzo[de]isoquinoline-5-sulfonate |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| CMA1 |
6-Chloro-1-methylindolin-2-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CMA1 |
(S)-2-[3-(4-Cyano-benzoylamino)-2,2-dimethyl-heptanoylamino]-3-phenyl-propionic acid ethyl ester |
NA |
510000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CMA1 |
6-Chloro-2,3-dihydro-1H-isoindol-1-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CMA1 |
Xeruborbactam |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| CMA1 |
Brintonamide A |
NA |
101000 |
NA |
NA |
NA |
NA |
TTD |
| CMA1 |
4-Chloro-1,3-dihydro-2H-indol-2-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CMA1 |
5-Chlorooxindole |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CMA1 |
(S)-ethyl 1-(5-(4-phenethoxybenzyl)-1,2,4-oxadiazol-3-yl)-6-amino-1-oxohexan-2-ylcarbamate |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CMA1 |
2-(1-Methoxy-ethylidene)-cyclopent-4-ene-1,3-dione |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CMA1 |
6-bromo-2,3-dihydro-1H-indol-2-one |
NA |
570000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| CMA1 |
2-Oxindole |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CMA1 |
7-Chloro-1,3-dihydro-2H-indol-2-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CMA1 |
4-Phenyl-2-phenylcarboxamidopentanoic anhydride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CMA1 |
2-(5,7-dichloro-3-hydroxy-2-oxo-1H-quinolin-4-yl)-2-oxoacetic acid |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB |
| CMA1 |
N-[(2S)-6-amino-1-[5-[[4-[2-(3,4-dichlorophenyl)ethoxy]phenyl]methyl]-1,2,4-oxadiazol-3-yl]-1-oxohexan-2-yl]-3,4-difluorobenzamide |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |