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      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CSNK2A1 N-(4-fluoro-1H-indazol-3-yl)-2,3-dihydro-1-benzofuran-5-carboxamide NA 200000 NA NA NA NA TTD
CSNK2A1 [(3,4-Dichlorophenyl)methyl][3-(dimethylamino)propyl]amine NA 1480000 NA NA NA NA BindingDB
CSNK2A1 N-((3,4-dichlorophenyl)methyl)cyclopropanamine NA 5000000 NA NA NA NA BindingDB
CSNK2A1 [(3,4-Dichlorophenyl)methyl](2-methylpropyl)amine NA 5000000 NA NA NA NA BindingDB
CSNK2A1 [(3,4-Dichlorophenyl)methyl](methyl)amine NA 750000 NA NA NA NA BindingDB
CSNK2A1 Benzenemethanamine, 3,4-dichloro-N-propyl- NA 1800000 NA NA NA NA BindingDB
CSNK2A1 4-[(3,4-Dichlorophenyl)methylamino]butan-1-ol NA 2390000 NA NA NA NA BindingDB
CSNK2A1 7-(hydroxymethyl)thieno[3,2-c]quinolin-4(5H)-one NA 8226000 NA NA NA NA BindingDB
CSNK2A1 4-Oxo-4,5-dihydrothieno[3,2-c]quinoline-7-carboxamide NA 8226000 NA NA NA NA BindingDB
CSNK2A1 Methyl 4-chlorothieno[3,2-c]quinoline-7-carboxylate NA 8226000 NA NA NA NA BindingDB
CSNK2A1 N-(3,4-dichlorobenzyl)-N-[3-(1H-imidazol-1-yl)propyl]amine NA 1900000 NA NA NA NA BindingDB
CSNK2A1 (3-Chloro-4-cyclopentyloxyphenyl)methanamine NA 5000000 NA NA NA NA BindingDB
CSNK2A1 3,4-Dichlorobenzoic acid NA 5000000 NA NA NA NA BindingDB
CSNK2A1 1-cyclohex-3-en-1-yl-N-[(3,4-dichlorophenyl)methyl]methanamine NA 3000000 NA NA NA NA BindingDB
CSNK2A1 N-[2-(p-Cinnamylamino)ethyl]-5-isoquinolone Sulfonamide 103900 NA NA NA NA NA BindingDB
CSNK2A1 Kinase inhibitor, A2 NA 131000 NA NA NA NA BindingDB
CSNK2A1 5-bromo-1H-indazole NA 410000 NA NA NA NA BindingDB|ChEMBL
CSNK2A1 2-[(4-oxo-5,5a,6,7,8,9,9a,9b-octahydro-3aH-thieno[3,2-c]quinoline-7-carbonyl)amino]benzoic acid NA 8226000 NA NA NA NA BindingDB
CSNK2A1 4-oxo-N-(pyridin-2-ylmethyl)-5,5a,6,7,8,9,9a,9b-octahydro-3aH-thieno[3,2-c]quinoline-7-carboxamide NA 8226000 NA NA NA NA BindingDB
CSNK2A1 4-oxo-N-(pyridin-3-ylmethyl)-5,5a,6,7,8,9,9a,9b-octahydro-3aH-thieno[3,2-c]quinoline-7-carboxamide NA 8226000 NA NA NA NA BindingDB