| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CSNK2A1 |
N-[4-[(1,1-dioxo-1,4-thiazinan-4-yl)methyl]phenyl]-4-oxo-5,5a,6,7,8,9,9a,9b-octahydro-3aH-thieno[3,2-c]quinoline-7-carboxamide |
NA |
8226000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSNK2A1 |
4-oxo-N-phenyl-5,5a,6,7,8,9,9a,9b-octahydro-3aH-thieno[3,2-c]quinoline-7-carboxamide |
NA |
8226000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSNK2A1 |
4-oxo-N-(2-phenylethyl)-5,5a,6,7,8,9,9a,9b-octahydro-3aH-thieno[3,2-c]quinoline-7-carboxamide |
NA |
8226000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSNK2A1 |
4-oxo-N-(pyridin-4-ylmethyl)-5,5a,6,7,8,9,9a,9b-octahydro-3aH-thieno[3,2-c]quinoline-7-carboxamide |
NA |
8226000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSNK2A1 |
N-benzyl-4-oxo-5,5a,6,7,8,9,9a,9b-octahydro-3aH-thieno[3,2-c]quinoline-7-carboxamide |
NA |
8226000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSNK2A1 |
4-[(3,4-Dichlorophenyl)methyl]morpholine |
NA |
5000000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSNK2A1 |
3,4-Dichlorophenylacetic acid |
NA |
5000000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSNK2A1 |
1-(3,4-Dichlorophenyl)pent-4-en-1-ol |
NA |
5000000 |
NA |
NA |
NA |
NA |
BindingDB |
| CSNK2A3 |
1-(2-Chlorobiphenyl-4-Yl)methanamine |
NA |
NA |
267000 |
NA |
NA |
NA |
BindingDB |
| CTBP2 |
Pyruvic Acid |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
| CTBP2 |
Hydrocinnamic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
| CTBP2 |
Phenylacetone |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
| CTBP2 |
Phenylpyruvic acid |
NA |
116300 |
NA |
NA |
NA |
NA |
PubChem |
| CTDSP1 |
(1,1-dioxo-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)-[4-(4-fluorophenyl)sulfonylpiperazin-1-yl]methanone |
NA |
219900 |
NA |
NA |
NA |
NA |
BindingDB |
| CTDSP1 |
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[4-(4-fluorophenyl)sulfonylpiperazin-1-yl]methanone |
NA |
797000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTH |
(2S,3R)-3-[(2S,3R)-5,7-dihydroxy-2-(4-methoxyphenyl)-4-oxo-2,3-dihydrochromen-3-yl]-5,7-dihydroxy-2-(4-hydroxyphenyl)-2,3-dihydrochromen-4-one |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| CTH |
8-[(2R,3S)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-2,3-dihydrochromen-3-yl]-7-hydroxy-2-(4-hydroxyphenyl)-5-methoxychromen-4-one |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| CTH |
Olsalazine |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| CTH |
Aurintricarboxylic Acid |
NA |
244500|282900|371100 |
NA |
NA |
NA |
NA |
BindingDB |
| CTH |
Salicylic Acid |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |