| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CTNNB1 |
4-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)butanenitrile |
120000|160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTNNB1 |
5-(2-(2H-Tetrazol-5-yl)ethyl)-5H-[1,2,5]oxadiazolo[3',4':5,6]pyrazino[2,3-b]indole |
NA|180000 |
770000|850000|NA |
NA |
NA |
NA |
NA |
BindingDB |
| CTNNB1 |
13-Oxa-10,12,14,16-tetrazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,8,10,14-heptaen-8-yldiazene |
230000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTNNB1 |
(4S)-5-anilino-4-[[(2S)-3-carboxy-2-[[(2S)-2-[(5-chloro-1H-indole-2-carbonyl)amino]-4-methylpentanoyl]amino]propanoyl]amino]-5-oxopentanoic acid |
NA |
273000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTNNB1 |
(4S)-4-[[(2S)-3-carboxy-2-[[(2S)-2-[(5-fluoro-1H-indole-2-carbonyl)amino]-3-naphthalen-2-ylpropanoyl]amino]propanoyl]amino]-5-methoxy-5-oxopentanoic acid |
NA |
349000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTNNB1 |
(4S)-4-[[(2S)-2-[[(2S)-2-[(4,6-dichloro-1H-indole-2-carbonyl)amino]-3-naphthalen-2-ylpropanoyl]amino]-3-(2H-tetrazol-5-yl)propanoyl]amino]-5-oxo-5-[4-(trifluoromethoxy)anilino]pentanoic acid |
173000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CTNNB1 |
2-((5-((4-ethylphenoxy)methyl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl)sulfanyl)cyclopentan-1-one |
NA |
NA |
580000 |
NA |
NA |
NA |
BindingDB |
| CTNNB1 |
Cercosporin, pure |
NA |
130000|150000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTNNB1 |
4-amino-N-isobutyl-1,2,5-oxadiazole-3-carboxamide |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTNNB1 |
4-Amino-1,2,5-oxadiazole-3-carboxamide |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTNNB1 |
Smer3 |
310000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTNNB1 |
|
240000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CTNNB1 |
2-(((2-(4-Ethylphenyl)-5-methyloxazol-4-yl)methyl)thio)-N-phenethylacetamide |
370000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTNNB1 |
Toxoflavin |
NA |
340000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTNNB1 |
(R)-Etodolac |
NA |
683000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| CTNNB1 |
4-(Pyrrolidine-1-carbonyl)-1,2,5-oxadiazol-3-amine |
1700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTNNB1 |
5H-[1,2,5]oxadiazolo[3',4':5,6]pyrazino[2,3-b]indole |
120000|280000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTNNB1 |
2-(9H-Indeno[1,2-B][1,2,5]oxadiazolo[3,4-E]pyrazin-9-yliden)-1-hydrazinecarbothioamide |
240000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTNNB1 |
1-Hydroxy-5-[2-(2H-tetrazol-5-yl)ethyl]-1H-indazole |
NA |
300000|350000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTNNB1 |
4-Amino-N-(phenylmethyl)-1,2,5-oxadiazole-3-carboxamide |
1700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |