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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CTNNB1 (S)-4-((S)-3-Carboxy-2-((S)-2-(2-(5-chloro-1H-indol-2-yl)acetamido)-3-(naphthalen-2-yl)propanamido)propanamido)-5-methoxy-5-oxopentanoic acid NA 210000|680000 NA NA NA NA BindingDB
CTRB1 Xeruborbactam NA 1000000 NA NA NA NA PubChem
CTRB2 Xeruborbactam NA 1000000 NA NA NA NA PubChem
CTRC {2-Oxo-1-[(3,3,3-trifluoro-1-isopropyl-2-oxo-propylcarbamoyl)-methyl]-1,2-dihydro-pyridin-3-yl}-carbamic acid benzyl ester 330000 NA NA NA NA NA BindingDB|TTD
CTRC N-[(2R)-3-(3-aminopropylsulfanyl)-1-[4-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-3,3-dimethyl-2,4-dihydro-1H-quinoline-8-sulfonamide 384000 NA NA NA NA NA BindingDB|TTD
CTRC 4-Phenyl-pyran-2-one 495000 NA NA NA NA NA BindingDB|TTD
CTRC 3,6-Bis[2-(4-bromo-2-sulfophenyl)diazenyl]-4,5-dihydroxy-2,7-naphthalenedisulfonic acid NA 110000 NA NA NA NA TTD
CTRC Phenol, 4-[2-(3-bromophenyl)diazenyl]- NA 220000 NA NA NA NA TTD
CTRC 3-Benzyl-6-bromo-pyran-2-one 112000 NA NA NA NA NA BindingDB|TTD
CTRC 6-Chloro-3-ethyl-pyran-2-one 785000 NA NA NA NA NA BindingDB|TTD
CTRC 6-Chloro-3-naphthalen-2-ylmethyl-pyran-2-one 625000 NA NA NA NA NA BindingDB|TTD
CTRC 3-Butyl-6-chloro-pyran-2-one 1980000 NA NA NA NA NA BindingDB|TTD
CTRC 6-Chloro-4-phenyl-pyran-2-one 382000 NA NA NA NA NA BindingDB|TTD
CTRC 3-Naphthalen-2-ylmethyl-pyran-2-one 267000 NA NA NA NA NA BindingDB|TTD
CTRC 3-Benzyl-6-trifluoromethyl-pyran-2-one 927000 NA NA NA NA NA BindingDB|TTD
CTRC 3-Naphthalen-1-ylmethyl-pyran-2-one 324000 NA NA NA NA NA BindingDB|TTD
CTRC 3-Benzyl-5-chloromethyl-pyran-2-one 412000 NA NA NA NA NA BindingDB|TTD
CTRC 3-Benzyl-5-trifluoromethyl-pyran-2-one 470000 NA NA NA NA NA BindingDB|TTD
CTRC 3-(4-Methoxy-benzyl)-5-trifluoromethyl-pyran-2-one 893000 NA NA NA NA NA BindingDB|TTD
CTRC 3-(4-Hydroxy-benzyl)-5-trifluoromethyl-pyran-2-one 1610000 NA NA NA NA NA BindingDB|TTD