| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CTRC |
3-Benzyl-pyran-2-one |
160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
3-Benzyl-5-bromo-pyran-2-one |
687000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
Xeruborbactam |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| CTRC |
N-{2-[(2-Acetylamino-propionyl)-hydrazono]-ethyl}-benzamide |
8000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTRC |
(8R,9S,13S,14S,17S)-3-methoxy-13-methyl-N-(3-phenylpropyl)-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-amine |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
4-[2-[(E)-2-(9-ethylcarbazol-3-yl)ethenyl]quinolin-1-ium-1-yl]butane-1-sulfonate |
NA |
NA |
351000 |
NA |
NA |
NA |
BindingDB |
| CTRC |
3-Fluoren-9-ylidenemethyl-piperidine |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
|
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTRC |
[3,5-Dibutyl-2-oxo-6-(6-oxoundecan-5-yl)pyran-4-yl] acetate |
190546|190546.07 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
[3,5-Dibutyl-2-oxo-6-(2-oxopropyl)pyran-4-yl] acetate |
660693|660693.45 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
[3,5-Dibutyl-2-(3-methyloxiran-2-yl)-6-oxopyran-4-yl] acetate |
501187|501187.23 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
[3,5-Dibutyl-2-(2-hydroxypropyl)-6-oxopyran-4-yl] acetate |
707946|707945.78 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
Bis(5-amidino-2-benzimidazolyl)methane |
120000|710000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CTRC |
5-Benzyl-pyran-2-one |
295000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
2-Chloro-benzenesulfonic acid 3-(3-guanidino-propoxy)-5-methyl-phenyl ester |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTRC |
|
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTRC |
4-Hydroxy-6-methyl-2-pyrone |
6309573|6309573.44 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
Elasnin |
223872|223872.11 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
4-Hydroxy-3,6-dimethyl-2H-pyran-2-one |
3467369|3467368.5 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTRC |
4-Hydroxy-3,5,6-trimethyl-2H-pyran-2-one |
1819701|1819700.86 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |