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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CTRC 4-Hydroxy-6-(2-oxo-2-phenylethyl)-2H-pyran-2-one 549541|549540.87 NA NA NA NA NA BindingDB|TTD
CTRC 3,5-Dibutyl-4-hydroxy-6-methylpyran-2-one 1348963|1348962.88 NA NA NA NA NA BindingDB|TTD
CTRC 4-Hydroxy-3,5-dimethyl-6-phenacylpyran-2-one 691831|691830.97 NA NA NA NA NA BindingDB|TTD
CTRC 3,5-Dibutyl-4-hydroxy-6-(2-oxopropyl)pyran-2-one 8128305|8128305.16 NA NA NA NA NA BindingDB|TTD
CTRC 2-Butyl-2-(3,5-dibutyl-4-hydroxy-6-oxopyran-2-yl)octanal 134896|134896.29 NA NA NA NA NA BindingDB|TTD
CTRC 4-Hydroxy-3-methyl-6-phenacylpyran-2-one 512861|512861.38 NA NA NA NA NA BindingDB|TTD
CTRC 3,5-dibutyl-4-hydroxy-6-[(E)-1-phenylprop-1-enyl]pyran-2-one 323594|323593.66 NA NA NA NA NA BindingDB|TTD
CTRC 2-[(5Z)-5-[(2-fluoro-5-nitro-phenyl)methylene]-4-oxo-2-thioxo-thiazolidin-3-yl]acetic acid NA 200000 NA NA NA NA TTD
CTRC 9-ethyl-3-[(E)-2-(1-methylquinolin-1-ium-2-yl)ethenyl]carbazole NA NA 110000 NA NA NA BindingDB
CTRC 4-[2-[(E)-2-(2-phenyl-1H-indol-3-yl)ethenyl]quinolin-1-ium-1-yl]butane-1-sulfonate NA NA 190000 NA NA NA BindingDB
CTRC {5-[1-{3-[4''-(2-tert-Butoxycarbonylamino-ethylsulfamoyl)-biphenyl-4-sulfonylamino]-phenyl}-eth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-acetic acid ethyl ester NA 375000 NA NA NA NA BindingDB
CTRC 4-{[(2-{(4-Chloro-benzyl)-[2-(3-{1-[3-ethoxycarbonylmethyl-4-oxo-2-thioxo-thiazolidin-(5Z)-ylidene]-ethyl}-phenoxycarbonylamino)-4-methyl-pentanoyl]-amino}-ethyl)-amino-methyl]di-benzoic acid methyl ester NA 210000 NA NA NA NA BindingDB
CTRC ZD 0892 200000 NA NA NA NA NA BindingDB|TTD
CTRL Xeruborbactam NA 1000000 NA NA NA NA PubChem
CTRL ethyl (E,4S)-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-hydroxypropanoyl]amino]propanoyl]amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]-7-(dimethylamino)-7-oxohept-2-enoate NA 330000 NA NA NA NA BindingDB
CTRL Ac-Ser-Ala-Val-Leu-Leu-al NA 3000000 NA NA NA NA BindingDB
CTRL Ac-Ser-Ala-Val-Leu-Gly(tBu)-al NA 3000000 NA NA NA NA BindingDB
CTRL Ac-Ser-Ala-Val-Leu-Phe-al NA 2000000 NA NA NA NA BindingDB
CTSA trans-Epoxysuccinyl-L-leucylamido-(4-guanidino)butane NA 300000 NA NA NA NA TTD
CTSA Vaborbactam NA 1000000 NA NA NA NA PubChem|TTD