| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CTSB |
Cbz-Lys-Phe-Lys-NH2 |
1494000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSB |
benzyl N-[(2S)-1-[[(2S)-1,5-diamino-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]carbamate |
2460000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSB |
Cbz-Gln-Phe-Lys-NH2 |
3545000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSB |
Cbz-Leu-Phe-Lys-NH2 |
1185000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSB |
(R)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)-N-((1S,2S)-1-{(S)-1-[2-((R)-1-benzylcarbamoyl-butylcarbamoyl)-pyrrolidine-1-carbonyl]-2-methyl-propylcarbamoyl}-2-methyl-butyl)-succinamic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CTSB |
(S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)-N-((1S,2S)-2-methyl-1-{(S)-2-methyl-1-[2-((S)-3,3,4,4,4-pentafluoro-2-oxo-1-propyl-butylcarbamoyl)-pyrrolidine-1-carbonyl]-propylcarbamoyl}-butyl)-succinamic acid |
NA |
416000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSB |
Cbz-Tyr-Lys-NH2 |
135000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSB |
Cbz-Phe-Lys(Me)-NH2 |
1547000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSB |
(R)-2-{[1-((S)-2-{(2S,3S)-2-[(R)-2-((S)-2-Acetylamino-3-carboxy-propionylamino)-3-carboxy-propionylamino]-3-methyl-pentanoylamino}-3-methyl-butyryl)-pyrrolidine-2-carbonyl]-amino}-pentanoic acid benzyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CTSB |
2-(Morpholin-4-ylmethyl)-4-nitrophenol |
212000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CTSB |
8-Hydroxy-5-nitroquinoline-2-carbonitrile |
123000|142000|214000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CTSB |
(1R,5R,7S)-3-benzoyl-6,6-dimethyl-1,7-bis(3-methylbut-2-enyl)bicyclo[3.3.1]nonane-2,4,9-trione |
NA |
103500 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSB |
[(S)-1-((S)-3-Methoxy-2-oxo-1-phenethyl-propylcarbamoyl)-3-methyl-butyl]-carbamic acid benzyl ester |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSB |
(2S,3S)-1,2-Epoxy-3-(Cbz-amino)-4-phenylbutane |
367000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CTSB |
(S)-N1-(2-Benzylcarbamoyl-1-methyl-2-oxoethyl)-2-[(S)-2-(3,3-dimethyl-butanoylamino)-3,3-dimethyl-butanoylamino]-N4,N4-dimethylsuccinamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| CTSC |
2-Amino-N-(1-benzyl-3-methanesulfonyl-allyl)-acetamide |
180000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSC |
4-(2-Amino-acetylamino)-5-phenyl-pent-2-enoic acid methyl ester |
220000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSC |
(2S)-2-[(2-aminoacetyl)amino]-3-phenylpropanamide |
6200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
N-[2-amino-3'-(3,6-dihydro-2H-pyran-4-yl)-1'-methoxyspiro[5,6-dihydro-1,3-oxazine-4,5'-chromeno[2,3-c]pyridine]-7'-yl]-5-chloropyridine-2-carboxamide |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
N-[2-amino-5'-fluoro-7'-(oxan-4-yl)spiro[5,6-dihydro-1,3-oxazine-4,9'-xanthene]-2'-yl]-5-methoxypyrazine-2-carboxamide |
NA |
378500 |
NA |
NA |
NA |
NA |
BindingDB |