| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CTSH |
8-(4-Methylpiperidin-1-yl)-5-nitroquinoline |
221000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSK |
[(S)-1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic acid (S)-2,2-dimethyl-1-(5-phenyl-[1,3,4]oxadiazol-2-ylmethyl)-propyl ester |
NA |
460000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSK |
tert-butyl N-[(1S)-2-phenyl-1-(prop-2-yn-1-ylcarbamoyl)ethyl]carbamate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSK |
tert-butyl N-{[(cyanomethyl)carbamoyl]methyl}carbamate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSK |
tert-butyl N-[(1S)-2-phenyl-1-(prop-2-en-1-ylcarbamoyl)ethyl]carbamate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSK |
Carbamic acid, [2-[(cyanomethyl)amino]-1-methyl-2-oxoethyl]-, 1,1-dimethylethyl ester, (s)- |
136000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSK |
benzyl N-{[(cyanomethyl)carbamoyl]methyl}carbamate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSK |
Cbz-Trp-Phe-Lys-NH2 |
639000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSK |
Cbz-Arg-Phe-Lys-NH2 |
147000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSK |
Cbz-Lys-Phe-Lys-NH2 |
284000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSK |
Cbz-Leu-Phe-Lys-NH2 |
213000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSL |
[(S)-1-(Isoxazol-5-ylmethyl)-aminooxalyl]-pentyl)-carbamic acid (S)-2,2-dimethyl-1-[3-(4-trifluoromethyl-phenyl)-pyrazol-1-ylmethyl]-propyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSL |
(1r)-1-{[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-2,2-dimethylpropyl(1S)-1-[oxo(1h-pyrazol-5-ylamino)acetyl]pentylcarbamate |
NA |
3800000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSL |
(1r)-2,2-dimethyl-1-({5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazol-2-yl}methyl)propyl(1S)-1-(oxo{[(1r)-1-phenylethyl]amino}acetyl)pentylcarbamate |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSL |
[(S)-1-(Pyridin-2-ylaminooxalyl)-pentyl]-carbamic acid (S)-2,2-dimethyl-1-[3-(4-trifluoromethyl-phenyl)-pyrazol-1-ylmethyl]-propyl ester |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSL |
[(S)-1-(Thiazol-2-ylaminooxalyl)-pentyl]-carbamic acid (S)-2,2-dimethyl-1-[4-(4-trifluoromethyl-phenyl)-imidazol-1-ylmethyl]-propyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSL |
(3S,3aS,6aR)-N-[1-(cyclopropylamino)-1,2-dioxohexan-3-yl]-2-[(2S)-3,3-dimethyl-2-[[(2S)-3-methyl-2-(pyrazine-2-carbonylamino)butanoyl]amino]butanoyl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole-3-carboxamide |
154000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSL |
Benzyl 1-((cyanomethyl)carbamoyl)cyclopentylcarbamate |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSL |
N-[1-(cyanomethylcarbamoyl)cyclohexyl]-4-(4-methylpiperazine-1-carbonyl)benzamide |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSL |
N-[1-(cyanomethylcarbamoyl)cyclohexyl]-4-[2-[4-(oxan-4-yl)piperazin-1-yl]-1,3-thiazol-4-yl]benzamide |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |