| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CTSG |
Acetyl-Ala-Ala-Pro-Ala-trifluromethane |
800000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSG |
4-N-[(2S)-3-methyl-1-oxo-1-[(2S)-2-[(5,5,6,6,6-pentafluoro-2-methyl-4-oxohexan-3-yl)carbamoyl]pyrrolidin-1-yl]butan-2-yl]-1-N-(4,4,4-trifluoro-3-oxo-1-phenylbutan-2-yl)benzene-1,4-dicarboxamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSG |
N-[(2S)-6-amino-1-[5-[[4-[2-(3,4-dichlorophenyl)ethoxy]phenyl]methyl]-1,2,4-oxadiazol-3-yl]-1-oxohexan-2-yl]-3,4-difluorobenzamide |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSG |
(2S,3S)-N-[(1R)-1-[[3-(butylamino)-3-oxopropyl]-diphenylsilyl]-3-methylbutyl]-3-methyl-2-[(2-naphthalen-2-ylacetyl)amino]pentanamide |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSG |
2-[(5-amino-1H-1,2,4-triazol-3-yl)sulfanyl]-N-(3,5-dichlorophenyl)-2-phenylacetamide |
NA |
139000 |
NA |
NA |
NA |
NA |
TTD |
| CTSG |
2,2',4-Trihydroxybenzophenone |
NA |
433200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSG |
5,5-Dimethyl-3-(4-methylphenyl)sulfonyl-1,3-oxazolidine-2,4-dione |
NA |
369000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSG |
6-Chloro-1,3-dihydroindol-2-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CTSG |
1-{2-[2-(5-Dimethylamino-naphthalene-1-sulfonylamino)-propionylamino]-propionyl}-pyrrolidine-2-carboxylic acid (3,3,3-trifluoro-1-isopropyl-2-oxo-propyl)-amide |
600000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSG |
2-{(S)-2-[((S)-1-{(S)-2-[4-(4-Chloro-benzenesulfonylaminocarbonyl)-benzoylamino]-3-methyl-butyryl}-pyrrolidine-2-carbonyl)-amino]-3-methyl-butyryl}-benzooxazole-5-carboxylic acid amide |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSH |
1-(2-Benzyloxycarbonylamino-propionyl)-aziridine-2,3-dicarboxylic acid diethyl ester |
160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSH |
3-(1-Benzyloxycarbonyl-3-methyl-butylcarbamoyl)-1-(2-tert-butoxycarbonylamino-3-phenyl-propionyl)-aziridine-2-carboxylic acid ethyl ester |
137000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSH |
1-((S)-2-tert-Butoxycarbonylamino-3-phenyl-propionyl)-aziridine-2,3-dicarboxylic acid diethyl ester |
210000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSH |
N-(1-cyanocyclopropyl)-8-hydroxy-5-nitroquinoline-7-carboxamide |
329000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSH |
N-(cyanomethyl)-8-hydroxy-5-nitroquinoline-7-carboxamide |
462000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSH |
N-[[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]methyl]-8-hydroxy-5-nitroquinoline-7-carboxamide |
108000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSH |
2-Bromo-4-nitronaphthalen-1-amine |
354000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSH |
Pyrrolidine, 1-(4-nitro-1-naphthalenyl)- |
251000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSH |
3-((S)-1-Benzyloxycarbonyl-3-methyl-butylcarbamoyl)-aziridine-2-carboxylic acid ethyl ester |
260000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSH |
2-[[(8-Hydroxy-5-nitroquinolin-7-yl)methyl]amino]acetonitrile |
129000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |