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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CYP2D6 (NZ)-N-[(5-pyridin-3-ylfuran-2-yl)methylidene]hydroxylamine NA 400000 NA NA NA NA TTD
CYP2D6 2-Fluoro-5-thiophen-3-yl-pyridine NA 199000 NA NA NA NA TTD
CYP2D6 2-Fluoro-5-(4-methyl-thiophen-3-yl)-pyridine NA 296000 NA NA NA NA TTD
CYP2D6 3-(1-Ethyl-1H-imidazol-4-yl)pyridine NA 344000 NA NA NA NA TTD
CYP2D6 rac-N,N-dimethyl-2-(3-(1-(thiazol-2-yl)ethyl)benzo[b]thiophen-2-yl)ethanamine NA 856000 NA NA NA NA TTD
CYP2D6 2,2-Dimethylbutyric acid NA 10000000 NA NA NA NA PubChem
CYP2D6 5-(3-{[1-(Benzylsulfonyl)piperidin-4-Yl]amino}phenyl)-4-Bromo-3-(Carboxymethoxy)thiophene-2-Carboxylic Acid NA 500000 NA NA NA NA TTD
CYP2D6 (-)-2-[2-(4-Chlorophenyl)benzyl]sulphinylacetamide NA 151000 NA NA NA NA TTD
CYP2D6 1-(3-Pyridin-3-ylisoxazol-5-YL)methanamine 400000 NA NA NA NA NA TTD
CYP2D6 3-Methyl-4-phenylthiophene 400000 NA NA NA NA NA TTD
CYP2D6 (5-Phenylthiophen-2-yl)methanamine 400000 NA NA NA NA NA TTD
CYP2D6 3-(4-Methyl-1,3-thiazol-2-yl)pyridine 400000 NA NA NA NA NA TTD
CYP2D6 N-[[(1S,5R)-3-(2-fluoro-2-methylpropyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide NA 734300 NA NA NA NA TTD
CYP2D6 N-[1-(cyclopropylmethyl)piperidin-4-yl]-3-propan-2-ylimidazo[1,5-a]pyridine-1-carboxamide NA 140100 NA NA NA NA TTD
CYP2D6 2-Amino-5-(3-aminopropyl)-6-phenyl-4-pyrimidinol NA 234000 NA NA NA NA TTD
CYP2D6 3-(Pyridin-3-yl)propan-1-amine 400000 NA NA NA NA NA TTD
CYP2D6 N-Salicylideneaniline NA 1000000 NA NA NA NA TTD
CYP2D6 6-(Pyridin-3-yl)-3,4-dihydroquinolin-2(1H)-one NA 171000 NA NA NA NA TTD
CYP2D6 1-[(2R)-1-hydroxy-3-phenylpropan-2-yl]-2-methylpyridin-1-ium-3,4-diol;chloride NA 200000 NA NA NA NA TTD
CYP2D6 6-Methoxyquinoline 1000000 NA NA NA NA NA TTD