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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CYP2D6 3-Quinuclidinol 1000000 NA NA NA NA NA TTD
CYP2D6 8-(1H-benzotriazol-1-ylamino)-octanoic acid NA 299000 NA NA NA NA TTD
CYP2D6 6-(Benzotriazol-1-ylamino)hexanoic acid NA 1710000 NA NA NA NA TTD
CYP2D6 1-(5-(Pyridin-3-yl)thiophen-2-yl)ethan-1-one NA 387000 NA NA NA NA TTD
CYP2D6 2-(4-Chlorophenyl)-3-hydroxy-8-phenylquinoline-4-carboxylic acid NA 151000 NA NA NA NA TTD
CYP2D6 [(2R)-1-(6-aminopurin-9-yl)propan-2-yl]oxymethyl-(3-hexadecylsulfanylpropoxy)phosphinate NA 110000 NA NA NA NA BindingDB
CYP2D6 2-[4-[2-Ethyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]piperidin-1-yl]-1-morpholin-4-ylethanone NA 133000 NA NA NA NA BindingDB
CYP2D6 3-(2-Methyl-1H-imidazol-1-yl)pyridine NA 277000 NA NA NA NA TTD
CYP2D6 Glycine, N-((5-((2-(4-chlorophenyl)-5-methyl-4-oxazolyl)methoxy)-2-fluorophenyl)methyl)-N-(methoxycarbonyl)- NA 150000 NA NA NA NA TTD
CYP2D6 5-Hydroxy saxagliptin NA 200000 NA NA NA NA TTD
CYP2D6 (5R)-3-[3-fluoro-4-(1-oxidotetrahydro-2H-thiopyran-4-yl)phenyl]-2-oxo-1,3-oxazolidine-5-carboxamide NA 900000 NA NA NA NA TTD
CYP2D6 (R)-1-(Methylsulfonylamino)-3-[2-(4-methoxyphenyl)ethyl]-4-(4-methoxy-phenyl)-2-imidazolidinone NA 180000 NA NA NA NA TTD
CYP2D6 1-[5-(6-Methoxynaphthalen-2-yl)pyridin-3-yl]ethanone NA 200000 NA NA NA NA TTD
CYP2D6 6-Pyridin-3-yl-3,4-dihydronaphthalen-2(1H)-one NA 171000 NA NA NA NA TTD
CYP2D6 1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)-4-(4-(trifluoromethyl)phenyl)pyridin-2(1H)-one NA 10000000 NA NA NA NA TTD
CYP2D6 4-(2,4-dichlorophenyl)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one NA 10000000 NA NA NA NA TTD
CYP2D6 4-((Benzylamino)methyl)benzoic acid NA 570000 NA NA NA NA TTD
CYP2D6 L-Chlorozotocin NA 2021000 NA NA NA NA PubChem|TTD
CYP2D6 4-(4-Phenylpiperidin-4-ylcarbonyl)morpholine hydrochloride NA 554000 NA NA NA NA TTD
CYP2D6 2-(2-Aminophenyl)quinazolin-4-amine NA 169000 NA NA NA NA TTD