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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CYP3A4 4-[[4-[2-[6-[2-(2,4-difluorophenyl)-1,1-difluoro-2-hydroxy-3-(tetrazol-1-yl)propyl]pyridin-3-yl]ethynyl]phenoxy]methyl]-N-methylbenzamide NA 122000 NA NA NA NA BindingDB|TTD
CYP3A4 2-(2,4-Difluorophenyl)-1,1-difluoro-1-[5-[2-[4-[(4-fluorophenyl)methoxy]phenyl]ethynyl]pyridin-2-yl]-3-(tetrazol-1-yl)propan-2-ol NA 200000 NA NA NA NA TTD
CYP3A4 Tert-Butyl {6-Oxo-6-[(Pyridin-3-Ylmethyl)amino]hexyl}carbamate NA NA 105000 NA NA NA BindingDB
CYP3A4 3-(1-Methylpyrrolidin-2-yl)pyridine NA 142400 NA NA NA NA BindingDB
CYP3A4 1-Naphthalenyl[4-(pentyloxy)-1-naphthalenyl]methanone NA 200000 NA NA NA NA PubChem|TTD
CYP3A5 2,2-Dimethylbutyric acid NA 10000000 NA NA NA NA PubChem
CYP3A7 Cinchophen NA NA NA NA 101490 NA PubChem
CYP51A1 Erythromycin NA 200000 NA NA NA NA PubChem|TTD
CYP51A1 Methimazole NA 200000 NA NA NA NA PubChem|TTD
CYP51A1 2-[(5-Chloro-1H-indole-2-carbonyl)-amino]-3-phenyl-propionic acid NA 200000 NA NA NA NA TTD
CYP51A1 Chlorpropamide NA 200000 NA NA NA NA PubChem|TTD
CYP51A1 Fluconazole NA NA|200000 120000|NA NA NA NA PubChem
CYP51A1 Metronidazole NA 200000 NA NA NA NA PubChem|TTD
CYP51A1 N-[1-(4-hydroxypiperidin-1-yl)-1-oxo-3-phenylpropan-2-yl]-1H-pyrrole-2-carboxamide NA 200000 NA NA NA NA TTD
CYP51A1 N-[(2S)-1-(4-hydroxypiperidin-1-yl)-1-oxo-3-phenylpropan-2-yl]-4,5,6,7-tetrahydro-1H-indole-2-carboxamide NA 200000 NA NA NA NA TTD
CYP51A1 Arachidonic Acid NA 200000 NA NA NA NA PubChem|TTD
CYP51A1 Propafenone NA 200000 NA NA NA NA PubChem|TTD
CYP51A1 Anandamide NA 200000 NA NA NA NA PubChem|TTD
CYP51A1 Lovastatin NA 200000 NA NA NA NA PubChem|TTD
CYP51A1 Sulfaphenazole NA 200000 NA NA NA NA PubChem|TTD