| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CYP51A1 |
Sulfinpyrazone |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| CYP51A1 |
Tolbutamide |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CYP51A1 |
Benzimidazole |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CYP51A1 |
Progesterone |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CYP51A1 |
Cholesterol |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CYP51A1 |
Pregnenolone |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CYTH2 |
N-(4-hydroxy-2,6-dimethylphenyl)-4-methoxybenzenesulfonamide |
1610000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| CYTH2 |
N-(4-hydroxy-3,5-dimethylphenyl)benzenesulfonamide |
5120000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| CYTH2 |
Cambridge id 7132364 |
540000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| CYTH2 |
N-(4-hydroxy-2-methylphenyl)-2,4,6-trimethylbenzenesulfonamide |
980000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| CYTH2 |
N-(4-hydroxy-2,6-dimethylphenyl)benzenesulfonamide |
NA|3720000 |
NA |
500000|NA|5e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| CYTH2 |
N-(4-hydroxy-2,6-dimethylphenyl)-4-methylbenzenesulfonamide |
1910000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| DAO |
3-Aminopyridine |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| DAO |
2-Amino-5-chlorobenzoic acid |
NA |
3929000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DAO |
3-Hydroxypicolinic Acid |
NA |
2478000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DAO |
3-Phenyl-4,5-dihydro-1,2,4-oxadiazol-5-one |
NA |
5000000 |
NA |
NA |
NA |
NA |
TTD |
| DAO |
7-Hydroxy-[1,2,4]triazolo[4,3-a]pyrimidine-6-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DAO |
6-(hydroxymethyl)-4-oxo-4H-pyran-3-yl 1H-pyrrole-2-carboxylate |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
| DAO |
2-[[2-[4-[2-[(Z)-[3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-ylidene]amino]oxyethyl]triazol-1-yl]acetyl]amino]-3-phenylpropanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DAO |
Oxiniacic Acid |
NA |
2500000 |
NA |
NA |
NA |
NA |
TTD |