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drugs and pathways
negative DTIs
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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
DDC
8-Methoxy-2,5-dimethylphenanthridin-5-ium;chloride
NA
600000
NA
NA
NA
NA
TTD
DDO
5-Fluoro-3-pyridinecarboxylic acid
NA
10000000
NA
NA
NA
NA
PubChem
DDO
3-Hydroxycoumarin
NA
7579000
NA
NA
NA
NA
BindingDB
DDO
6-Aminonicotinic acid
NA
2364000
NA
NA
NA
NA
BindingDB
DDO
5-(Methylamino)pyridine-3-carboxylic acid
NA
3541000
NA
NA
NA
NA
BindingDB
DDO
2-Amino-5-methylthiophene-3-carboxylic acid
NA
4251000
NA
NA
NA
NA
BindingDB
DDO
Benzoic Acid
NA
10000000
NA
NA
NA
NA
PubChem
DDO
5-Methylnicotinic acid
NA
5472000
NA
NA
NA
NA
BindingDB
DDO
5-Hydroxynicotinic acid
NA
3351000
NA
NA
NA
NA
BindingDB
DDO
5-Chloro-3-hydroxyquinolin-2(1H)-one
NA
206000
NA
NA
NA
NA
BindingDB
DDO
meso-Tartaric acid
NA
3922000
NA
NA
NA
NA
BindingDB
DDO
3'-Hydroxycinnamic acid
NA
10000000
NA
NA
NA
NA
PubChem
DDO
Malonic acid
NA|153000
879000|1355000|NA
NA
NA
NA
NA
BindingDB|PubChem
DDO
Nicotinic acid
NA
2778000
NA
NA
NA
NA
BindingDB|PubChem
DDO
5-Chlorosalicylic Acid
NA
10000000
NA
NA
NA
NA
PubChem
DDR1
N'-(5-chloro-2-ethylsulfonylphenyl)-2-methyl-6-oxopiperidine-4-carbohydrazide
NA
118800
NA
NA
NA
NA
BindingDB
DDR1
N-[(5-chloro-2-ethylsulfonylphenyl)methyl]-6-oxo-5-(trifluoromethyl)piperidine-3-carboxamide
NA
139800
NA
NA
NA
NA
BindingDB
DDX3X
3-[(5Z)-5-[(3-bromophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-(4-hydroxyphenyl)propanamide
NA
300000
NA
NA
NA
NA
BindingDB
DDX3X
2-(3-(5-(3-Bromobenzylidene)-4-oxo-2-thioxothiazolidin-3-yl)propanamido)benzoic acid
NA
200000
NA
NA
NA
NA
BindingDB
DDX3X
3-(5-(2-methoxybenzylidene)-4-oxo-2-thioxothiazolidin-3-yl)-N-(3-hydroxyphenyl)propanamide
NA
200000
NA
NA
NA
NA
BindingDB
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