| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DDX3X |
4-(5-(3-bromobenzylidene)-4-oxo-2-thioxothiazolidin-3-yl)-N-(3-hydroxyphenyl)butanamide |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| DDX3X |
4-(5-(3-bromobenzylidene)-4-oxo-2-thioxothiazolidin-3-yl)-N-(2-hydroxyphenyl)butanamide |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB |
| DDX3X |
5-amino-3-(1-cyano-2-(5-(2-nitrophenyl)furan-2-yl)vinyl)-1-phenyl-1H-pyrazole-4-carbonitrile |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
| DDX3X |
5-amino-3-[(Z)-2-[5-(3-chlorophenyl)furan-2-yl]-1-cyanoethenyl]-1-phenylpyrazole-4-carbonitrile |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGAT1 |
{4-[4-(6-Carbamoyl-3,5-dimethylpyrazin-2-yl)phenyl]cyclohexyl}acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
| DGAT2 |
{4-[4-(6-Carbamoyl-3,5-dimethylpyrazin-2-yl)phenyl]cyclohexyl}acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
| DGKA |
US11964973, Example 383 |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKA |
US11964973, Example 318 |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKA |
US11964973, Example 324 |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 17 |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 30 |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 11 |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 37 |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 42 |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 47 |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 13 |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 236 |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 29 |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 3 |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB |
| DGKZ |
US11964973, Example 185 |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |