| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DGKZ |
US11964973, Example 382 |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
5-(1,3,4,9-Tetrahydro-beta-carbolin-2-ylmethyl)-pyrimidine-2,4-diamine |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
2-Amino-6,7-dimethyl-3,7-dihydropyrimido[4,5-b][1,4]oxazin-4-one |
NA |
377000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHFR |
2-Amino-6-methyl-3,7-dihydropyrimido[4,5-b][1,4]oxazin-4-one |
NA |
242000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHFR |
2-Amino-6-methyl-7-phenyl-3,7-dihydropyrimido[4,5-b][1,4]oxazin-4-one |
NA |
740000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHFR |
6,7-Dimethyl-7H-pyrimido[4,5-b][1,4]oxazine-2,4-diamine |
NA |
903000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHFR |
6-phenyl-7H-pyrimido[4,5-b][1,4]oxazine-2,4-diamine |
NA |
168000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHFR |
5-Methyluridine 5'-(dihydrogen phosphate) |
NA |
340000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
(2S)-2-{[4-({2-amino-5-methyl-4-oxo-3H,4H,7H-pyrrolo[2,3-d]pyrimidin-6-yl}sulfanyl)phenyl]formamido}pentanedioic acid |
NA |
240000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
2-{4-[(2-Amino-4-oxo-3,4,5,6,7,8-hexahydro-pyrido[2,3-d]pyrimidin-6-ylmethyl)-amino]-benzoylamino}-4-phosphono-butyric acid |
NA |
220000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
2-[[4-[[(2-amino-4-oxo-5,6,7,8-tetrahydro-3H-pyrido[2,3-d]pyrimidin-6-yl)amino]methyl]benzoyl]amino]pentanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
2-[[4-[[(2-amino-4-oxo-5,6,7,8-tetrahydro-3H-pyrido[2,3-d]pyrimidin-6-yl)-methylamino]methyl]benzoyl]amino]pentanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
2-{4-[(2-Amino-4-oxo-3,4,5,6,7,8-hexahydro-pyrido[2,3-d]pyrimidin-6-ylmethyl)-amino]-benzoylamino}-4-(ethoxy-hydroxy-phosphoryl)-butyric acid |
NA |
950000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
5-(((2-Methylpyridin-3-yl)oxy)methyl)quinazoline-2,4-diamine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
Mtb-DHFR inhibitor IND-07 |
NA |
980000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHFR |
Mtb-DHFR inhibitor KC-11 |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHFR |
1-[1-Benzyl-5-[[1-(3-chlorophenyl)triazol-4-yl]methoxy]-2-methylindol-3-yl]ethanone |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHFR |
Naproxen |
7000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| DHFR |
(7S)-N,N-dipropyl-5,6,7,8-tetrahydroindolizin-7-amine |
NA |
325000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
|
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |