| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DHFR |
|
NA |
950000 |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
1,1-Bis(4-hydroxyphenyl)benzo[e]isobenzofuran-3-one |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHFR |
3,3-Bis(3-fluoro-4-hydroxy-phenyl)benzo[g]isobenzofuran-1-one |
109000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DHFR |
4-(4,6-diamino-2,2-dimethyl-1,3,5-triazin-1(2H)-yl)benzenesulfonamide |
154882 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
1-[3-(2,5-Dimethylanilino)propoxy]-6,6-dimethyl-1,3,5-triazine-2,4-diamine;hydrobromide |
124000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
1-[3-(4-chlorophenoxy)propoxy]-2-methyl-2H-1,3,5-triazine-4,6-diamine;hydrobromide |
116000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
1-[3-(Diethylamino)propoxy]-6,6-dimethyl-1,3,5-triazine-2,4-diamine;hydrobromide |
230000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
2-phenyl-1-[3-(2,4,5-trichlorophenoxy)propoxy]-2H-1,3,5-triazine-4,6-diamine;hydrobromide |
145000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
Naproxen, (-)- |
3400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
N-(4-Aminobenzoyl)-L-glutamic acid |
180000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
Iclaprim |
NA |
300000 |
NA |
NA |
NA |
NA |
PubChem |
| DHFR |
5-{[1-(2-Fluorobenzyl)piperidin-4-yl]methoxy}quinazoline-2,4-diamine |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
(2-Chlorophenyl)-[4-(2,4-diaminoquinazolin-5-yloxymethyl)piperidin-1-yl]methanone |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
5-((1-(2-Fluorophenylsulfonyl)piperidin-4-yl)methoxy)quinazoline-2,4-diamine |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
(3-Chlorophenyl)(4-((2,4-diaminoquinazolin-5-yloxy)methyl)piperidin-1-yl)methanone |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| DHFR |
Diclofenac |
160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| DHFR |
Ethyl 4-(4,6-diamino-2,2-dimethyl-1,3,5-triazin-1-yl)benzoate |
346737 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
4-(4,6-Diamino-2,2-dimethyl-1,3,5-triazin-1-yl)benzonitrile |
204174 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DHFR |
Etodolac |
1800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| DHFR |
Fenbufen |
360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |